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Items 1 to 401 of 401 total
 Nocodazole, Microtubule Inhibitor / CRISPR Editing Enhancer Nocodazole, Microtubule Inhibitor / CRISPR Editing Enhancer
Nocodazole, Microtubule Inhibitor / CRISPR Editing Enhancer
$79.00 
Catalog No. M60331
A potent microtubule inhibitor to inhibit mitosis and CRISPR editing enhancer.
(+)-JQ1, BET Inhibitor(+)-JQ1, BET Inhibitor
(+)-JQ1, BET Inhibitor
$109.00   $139.00 
Catalog No. M60139
A potent and selective inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3, and BRD4
(R)-2-HG， a-KG-dependent dioxygenases inhibitor (R)-2-HG， a-KG-dependent dioxygenases inhibitor 
(R)-2-HG， a-KG-dependent dioxygenases inhibitor
$69.00 
Catalog No. M60104
An a-KG-dependent dioxygenases inhibitor
(S)-crizotinib, MTH1 Inhibitor(S)-crizotinib, MTH1 Inhibitor
(S)-crizotinib, MTH1 Inhibitor
$99.00 
Catalog No. M60208
A novel potent, selective and cell permeable MTH1 inhibitor.
(Z)-4-Hydroxytamoxifen, CRISPR Editing Enhancer(Z)-4-Hydroxytamoxifen, CRISPR Editing Enhancer
(Z)-4-Hydroxytamoxifen, CRISPR Editing Enhancer
$89.00 
Catalog No. M60324
Previously characterized as an Estrogen Receptor antagonist and now found to improve genome-editing specificity in CRISPR-mediated gene editing
1,4-DPCA, Prolyl 4-hydroxylase (P4H) Inhibitor1,4-DPCA, Prolyl 4-hydroxylase (P4H) Inhibitor
1,4-DPCA, Prolyl 4-hydroxylase (P4H) Inhibitor
$29.00 
Catalog No. M60288
A selective and cell permeable prolyl 4-hydroxylase (P4H) inhibitor.
1-methyl-D-tryptophan (D-1MT), IDO Inhibitor1-methyl-D-tryptophan (D-1MT), IDO Inhibitor
1-methyl-D-tryptophan (D-1MT), IDO Inhibitor
$29.00 
Catalog No. M60291
A potent and selective indoleamine 2,3-dioxygenase (IDO) inhibitor.
4SC-202, HDAC/LSD1 Dual Inhibitor 4SC-202, HDAC/LSD1 Dual Inhibitor 
4SC-202, HDAC/LSD1 Dual Inhibitor
$109.00 
Catalog No. M60230
A potent, selective and orally bioavailable HDAC/LSD1 dual Inhibitor.
5-Azacytidine, DNA Methyltransferase Inhibitor5-Azacytidine, DNA Methyltransferase Inhibitor
5-Azacytidine, DNA Methyltransferase Inhibitor
$59.00 
Catalog No. M60131
A classic DNA methyltransferase inhibitor, incorporates into DNA forming covalent adducts with cellular DNMT, depleting enzyme activity.
A-366, G9a/GLP HMTase InhibitorA-366, G9a/GLP HMTase Inhibitor
A-366, G9a/GLP HMTase Inhibitor
$139.00 
Catalog No. M60210
A novel highly potent, selective and cell permeable G9a/GLP histone lysine methyltransferase inhibitor.
A01, Smurf1 E3 Ubiquitin Ligase InhibitorA01, Smurf1 E3 Ubiquitin Ligase Inhibitor
A01, Smurf1 E3 Ubiquitin Ligase Inhibitor
$109.00 
Catalog No. M60249
A potent and selective Smurf1 E3 ubiquitin ligase inhibitor.
A769662, AMPK ActivatorA769662, AMPK Activator
A769662, AMPK Activator
$79.00 
Catalog No. M60020
A potent allosteric AMPK activator.
A83-01, TGF-β Inhibitor A83-01, TGF-β Inhibitor 
A83-01, TGF-β Inhibitor
$59.00 
Catalog No. M60021
A potent and selective TGF-β pathway inhibitor (targeting ALK4, ALK5 and ALK7).
AA92593, Antagonist of Melanopsin-mediated Photo-transductionAA92593, Antagonist of Melanopsin-mediated Photo-transduction
AA92593, Antagonist of Melanopsin-mediated Photo-transduction
$139.00 
Catalog No. M60143
A potent and selective small molecule antagonist of melanopsin-mediated photo-transduction.
Abiraterone, CYP17 inhibitor Abiraterone (CB-7598)Abiraterone, CYP17 inhibitor Abiraterone (CB-7598)
Abiraterone, CYP17 inhibitor Abiraterone (CB-7598)
$69.00 
Catalog No. M60031
A first-in-class CYP17 inhibitor approved to treat castration-resistant prostate cancer.
ABT-199, BCL-2 inhibitorABT-199, BCL-2 inhibitor
ABT-199, BCL-2 inhibitor
$99.00 
Catalog No. M60075
A potent BCL-2–selective (BCL-X L) inhibitor with clinical efficacy.
ACY-1215 (Rocilinostat), HDAC6 inhibitorACY-1215 (Rocilinostat), HDAC6 inhibitor
ACY-1215 (Rocilinostat), HDAC6 inhibitor
$109.00 
Catalog No. M60076
A highly potent, selective, and orally bioavailable inhibitor of histone deacetylase 6 (HDAC6).
ADC Toxin Monomethyl auristatin E (MMAE)ADC Toxin Monomethyl auristatin E (MMAE)
ADC Toxin Monomethyl auristatin E (MMAE)
Inquiry 
Catalog No. T60001
Antimitotic agent used as toxin linked to antibody.
ADC Toxin Monomethyl auristatin F (MMAF)ADC Toxin Monomethyl auristatin F (MMAF)
ADC Toxin Monomethyl auristatin F (MMAF)
Inquiry   xcessbio新品中国*代理
Catalog No. T60002
Antimitotic agent used as toxin linked to antibody
AdipoRon, Adiponectin Receptor/AdipoR agonist AdipoRon, Adiponectin Receptor/AdipoR agonist 
AdipoRon, Adiponectin Receptor/AdipoR agonist
$129.00 
Catalog No. M60152
A novel, highly potent, selective and orally active small molecule agonist of adiponectin receptor (AdipoR).
AG-120 (Ivosidenib), IDH1 InhibitorAG-120 (Ivosidenib), IDH1 Inhibitor
AG-120 (Ivosidenib), IDH1 Inhibitor
$129.00 
Catalog No. M60318
A potent, selective and reversible inhibitor of IDH1 in clinical trials.
AG-221 (Enasidenib), IHD2 InhibitorAG-221 (Enasidenib), IHD2 Inhibitor
AG-221 (Enasidenib), IHD2 Inhibitor
$129.00 
Catalog No. M60296
A potent and selective inhibitor of IDH2 R140Q mutant.
AGI-5198 (IDH-C35), Mutant IDH1 Inhibitor AGI-5198 (IDH-C35), Mutant IDH1 Inhibitor 
AGI-5198 (IDH-C35), Mutant IDH1 Inhibitor
$109.00 
Catalog No. M60068
The first highly potent and selective mutant IDH1 inhibitor that was shown to have anti-tumor efficacy in vivo.
AGI-6780, Mutant IDH2 Inhibitor AGI-6780, Mutant IDH2 Inhibitor 
AGI-6780, Mutant IDH2 Inhibitor
$109.00 
Catalog No. M60105
The first highly potent and selective small molecule mutant IDH2 inhibitor.
AK-7, SIRT2 InhibitorAK-7, SIRT2 Inhibitor
AK-7, SIRT2 Inhibitor
$69.00 
Catalog No. M60107
A cell- and brain-permeable, selective sirtuin SIRT2 inhibitor, displays no effect on SIRT1 or SIRT3.
AMI-1, Histone Methyltransferase InhibitorAMI-1, Histone Methyltransferase Inhibitor
AMI-1, Histone Methyltransferase Inhibitor
$79.00 
Catalog No. M60272
A potent and specific small molecule inhibitor of histone methyltransferase targeting yeast Hmt1p and human PRMT1.
APY29, IRE1a Modulator APY29, IRE1a Modulator 
APY29, IRE1a Modulator
$109.00 
Catalog No. M60168
A highly potent and selective small molecule modulator of IRE1α.
AR7, RARα antagonist AR7, RARα antagonist 
AR7, RARα antagonist
$129.00 
Catalog No. M60116
A highly potent and selective enhancer of the chaperone-mediated autophagy (CMA) through antagonizing RARα.
AS2034178, GPR40 Agonist AS2034178, GPR40 Agonist 
AS2034178, GPR40 Agonist
$139.00 
Catalog No. M60221
A potent, selective and orally bioavailable GPR40 (FFA1) agonist.
AS8351, KDM5B InhibitorAS8351, KDM5B Inhibitor
AS8351, KDM5B Inhibitor
$109.00 
Catalog No. M60330
A potent iron chelator that has been found to inhibit of histone demethylase KDM5B (JARID1B).
Atglistatin, Adipose Triglyceride Lipase (ATGL) Inhibitor Atglistatin, Adipose Triglyceride Lipase (ATGL) Inhibitor 
Atglistatin, Adipose Triglyceride Lipase (ATGL) Inhibitor
$119.00 
Catalog No. M60150
A highly potent, selective and competitive inhibitor of adipose triglyceride lipase (ATGL).
AZD2014, mTOR InhibitorAZD2014, mTOR Inhibitor
AZD2014, mTOR Inhibitor
$169.00 
Catalog No. M60090
A highly potent, selective and ATP-competitive mTOR inhibitor with a high level of selectivity against other members of the PIKK family.
AZD6244 (Selumetinib), MEK Inhibitor AZD6244 (Selumetinib), MEK Inhibitor 
AZD6244 (Selumetinib), MEK Inhibitor
$109.00 
Catalog No. M60067
A potent and highly selective non-ATP competitive MEK inhibitor in clinical trials.
AZD8055, mTOR InhibitorAZD8055, mTOR Inhibitor
AZD8055, mTOR Inhibitor
$69.00 
Catalog No. M60091
A highly potent, selective and ATP-competitive mTOR inhibitor with >1,000-fold selectivity against all PI3K isoforms.
Azidothymidine (AZT), Reverse Transcriptase Inhibitor Azidothymidine (AZT), Reverse Transcriptase Inhibitor 
Azidothymidine (AZT), Reverse Transcriptase Inhibitor
$29.00 
Catalog No. M60238
A selective, orally bioavailable and brain penetrant| reverse transcriptase inhibitor.
b-AP15 (NSC687852), Deubiquitinases Inhibitorb-AP15 (NSC687852), Deubiquitinases Inhibitor
b-AP15 (NSC687852), Deubiquitinases Inhibitor
$89.00 
Catalog No. M60251
A potent and selective deubiquitinases inhibitor for 19S proteasomes activity of Ub-AMC cleavage.
BAF312, S1P1/5 Selective AgonistBAF312, S1P1/5 Selective Agonist
BAF312, S1P1/5 Selective Agonist
$129.00 
Catalog No. M60039
A potent and selective sphingosine 1-phosphate (S1P1/5) receptor agonist in clinical trials.
BAM7, BAX ActivatorBAM7, BAX Activator
BAM7, BAX Activator
$109.00 
Catalog No. M60069
The first potent and selective small molecule activator of BAX, which is a pro-apoptotic BCL-2 family member.
BAY 87-2243, Hypoxia-inducible Factor-1 (HIF-1) InhibitorBAY 87-2243, Hypoxia-inducible Factor-1 (HIF-1) Inhibitor
BAY 87-2243, Hypoxia-inducible Factor-1 (HIF-1) Inhibitor
$119.00 
Catalog No. M60217
A highly potent and selective hypoxia-inducible factor-1 (HIF-1) inhibitor.
BAY11-7082, E2 Ubiquitin Conjugating Enzyme InhibitorBAY11-7082, E2 Ubiquitin Conjugating Enzyme Inhibitor
BAY11-7082, E2 Ubiquitin Conjugating Enzyme Inhibitor
$89.00 
Catalog No. M60309
A potent and selective E2 ubiquitin (Ub) conjugating enzyme inhibitor.
BAZ2-ICR, BAZ2 Bromodomain InhibitorBAZ2-ICR, BAZ2 Bromodomain Inhibitor
BAZ2-ICR, BAZ2 Bromodomain Inhibitor
$129.00 
Catalog No. M60226
A potent and selective BAZ2 bromodomain inhibitor.
BETP, GLP-1R PotentiatorBETP, GLP-1R Potentiator
BETP, GLP-1R Potentiator
$129.00 
Catalog No. M60196
A positive allosteric modulator and partial agonist of the glucagon-like peptide 1 (GLP-1) receptor.
BG45, HDAC3 InhibitorBG45, HDAC3 Inhibitor
BG45, HDAC3 Inhibitor
$59.00 
Catalog No. M60266
A potent, selective and cell permeable HDAC3 inhibitor.
BI-2536, PLK1 and BRD4 Dual Inhibitor BI-2536, PLK1 and BRD4 Dual Inhibitor 
BI-2536, PLK1 and BRD4 Dual Inhibitor
$119.00 
Catalog No. M60171
BI-2536 is a potent inhibitor of PLK1 (Polo-like kinase 1) and BRD4 in clinical trials.
BI-7273, BRD9 Bromodomain InhibitorBI-7273, BRD9 Bromodomain Inhibitor
BI-7273, BRD9 Bromodomain Inhibitor
$129.00 
Catalog No. M60322
A potent, selective and cell-permeable BRD9 inhibitor.
BI-9564, BRD9 Bromodomain InhibitorBI-9564, BRD9 Bromodomain Inhibitor
BI-9564, BRD9 Bromodomain Inhibitor
$129.00 
Catalog No. M60323
A potent, selective and cell-permeable BRD9 inhibitor.
BIBW2992(Afatinib), EGFR Inhibitor BIBW2992(Afatinib), EGFR Inhibitor 
BIBW2992(Afatinib), EGFR Inhibitor
$109.00 
Catalog No. M60065-5s
A potent and selective irreversible inhibitor of EGFR/HER2 in clinical trials.
Bioymifi, TRAIL Receptor DR5 ActivatorBioymifi, TRAIL Receptor DR5 Activator
Bioymifi, TRAIL Receptor DR5 Activator
$109.00 
Catalog No. M60088
A potent and selective small molecule agonist of DR5.
BIX-01294, G9a/GLP HMTase InhibitorBIX-01294, G9a/GLP HMTase Inhibitor
BIX-01294, G9a/GLP HMTase Inhibitor
$79.00 
Catalog No. M60216
A potent and selective G9a and GLP histone lysine methyltransferase inhibitor.
BMI1 Mouse Monoclonal AntibodyBMI1 Mouse Monoclonal Antibody
BMI1 Mouse Monoclonal Antibody
$0.00 
Catalog No. A90010-5
BMI1 Mouse Monoclonal Antibody.
BMS-708163 (Avagacestat), γ-Secretase InhibitorBMS-708163 (Avagacestat), γ-Secretase Inhibitor
BMS-708163 (Avagacestat), γ-Secretase Inhibitor
$89.00 
Catalog No. M60032
A potent γ-secretase Inhibitor, more selective for APP than Notch, in clinical trials for Alzheimer's disease.
BQU57, GTPase Ral InhibitorBQU57, GTPase Ral Inhibitor
BQU57, GTPase Ral Inhibitor
$139.00 
Catalog No. M60228
A potent and selective GTPase Ral Inhibitor
BRD9757, HDAC6 InhibitorBRD9757, HDAC6 Inhibitor
BRD9757, HDAC6 Inhibitor
$129.00 
Catalog No. M60117
A highly potent and selective HDAC6 inhibitor.
Bromosporine, Pan-bromodomain InhibitorBromosporine, Pan-bromodomain Inhibitor
Bromosporine, Pan-bromodomain Inhibitor
$129.00 
Catalog No. M60144
A broad spectrum inhibitor for bromodomains.
C646, p300/CBP inhibitorC646, p300/CBP inhibitor
C646, p300/CBP inhibitor
$129.00 
Catalog No. M60129
A potent, selective and cell-permeable p300/CBP histone acetyltransferase (HAT) inhibitor.
Carfilzomib, Proteasome InhibitorCarfilzomib, Proteasome Inhibitor
Carfilzomib, Proteasome Inhibitor
$109.00 
Catalog No. M60109
A selective, irreversible proteasome inhibitor.
CASIN, Cdc42 Inhibitor CASIN, Cdc42 Inhibitor 
CASIN, Cdc42 Inhibitor
$139.00 
Catalog No. M60040
A novel and potent inhibitor of Cdc42; was shown to rescue HSC aging phenotype and promote HSC transplantation efficiency.
CAY10603, HDAC6 InhibitorCAY10603, HDAC6 Inhibitor
CAY10603, HDAC6 Inhibitor
$129.00 
Catalog No. M60234
A potent and selective HDAC6 inhibitor.
CB-5083, p97 AAA ATPase Inhibitor CB-5083, p97 AAA ATPase Inhibitor 
CB-5083, p97 AAA ATPase Inhibitor
$129.00 
Catalog No. M60306
A highly potent, selective and orally bioavailable p97 AAA ATPase inhibitor.
CBX5 Polyclonal AntibodyCBX5 Polyclonal Antibody
CBX5 Polyclonal Antibody
$0.00 
Catalog No. A70033
Chromobox protein homolog 5
CHIR99021, GSK3β Inhibitor CHIR99021, GSK3β Inhibitor 
CHIR99021, GSK3β Inhibitor
$390.00 
Catalog No. M60002  xcessbio新品中国*代理
The most widely used, potent and selective GSK3β Inhibitor; Wnt pathway activator.
CI994 (Tacedinaline), HDAC InhibitorCI994 (Tacedinaline), HDAC Inhibitor
CI994 (Tacedinaline), HDAC Inhibitor
$59.00 
Catalog No. M60186
A potent, selective and orally active histone deacetylase (HDAC) inhibitor targeting HDAC1, HDAC2 and HDAC3.
Cilliobrevin D, AAA+ ATPase Motor Cytoplasmic Dynein Inhibitor Cilliobrevin D, AAA+ ATPase Motor Cytoplasmic Dynein Inhibitor 
Cilliobrevin D, AAA+ ATPase Motor Cytoplasmic Dynein Inhibitor
$139.00 
Catalog No. M60041-2s
A novel and specific inhibitor of the AAA+ ATPase motor cytoplasmic dynein; perturbs protein| trafficking within the primary cilium and affects other dynein-dependent processes, such as spindle pole focusing, kinetochore-microtubule attachment, melanosome aggregation and peroxisome motility in cultured cells.
Compound Library of Bromodomain/BETCompound Library of Bromodomain/BET
Compound Library of Bromodomain/BET
$1150.00   $1437.00 
Catalog No. LI30006
Compound Library of Bromodomain/BET set is composed of 23 small molecules in separated vials.
Compound Library of HDACCompound Library of HDAC
Compound Library of HDAC
$700.00   $850.00 
Catalog No. LI30005
Compound Library of HDAC set is composed of 18 small molecules in separated vials.
Compound Library of Histone DemethylaseCompound Library of Histone Demethylase
Compound Library of Histone Demethylase
$1400.00 
Catalog No. LI30003
Library of Histone Demethylase is composed of 15 small molecules in separated vials.
Compound Library of Histone MethyltransferaseCompound Library of Histone Methyltransferase
Compound Library of Histone Methyltransferase
$1200.00 
Catalog No. LI30002
Compound Library of Histone Methyltransferase is composed of 14 small molecules in separated vials.
Compound Library of Hypoxia Inducible FactorCompound Library of Hypoxia Inducible Factor
Compound Library of Hypoxia Inducible Factor
$360.00   $446.00 
Catalog No. LI30007
Epigenetic compounds library of Hypoxia Inducible Factor
CP-690550, JAK InhibitorCP-690550, JAK Inhibitor
CP-690550, JAK Inhibitor
$79.00 
Catalog No. M60033
A potent and selective pan-JAK Inhibitor in clinical trials for rheumatoid arthritis.
CPI-169, EZH2 Methyltransferase InhibitorCPI-169, EZH2 Methyltransferase Inhibitor
CPI-169, EZH2 Methyltransferase Inhibitor
$129.00 
Catalog No. M60275
A highly potent and selective small molecule inhibitor of histone methyltransferase EZH2.
CPI-455, KDM5 Demethylases Inhibitor CPI-455, KDM5 Demethylases Inhibitor 
CPI-455, KDM5 Demethylases Inhibitor
$129.00 
Catalog No. M60326
A potent and selective KDM inhibitor.
CPI203, BET InhibitorCPI203, BET Inhibitor
CPI203, BET Inhibitor
$139.00 
Catalog No. M60124
A novel potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4, inhibiting Myc expression.
CRISPR Editing Tool BoxCRISPR Editing Tool Box
CRISPR Editing Tool Box
$499.00 
Catalog No. LI30010
Compound collection for CRISPR editing.
CTEP, mGlu5 AntagonistCTEP, mGlu5 Antagonist
CTEP, mGlu5 Antagonist
$259.00 
Catalog No. M60099
A highly potent, selective and orally bioavailable allosteric antagonist of mGlu5 receptor.
CUDC-101， HDAC/EGFR/HER2 Inhibitor CUDC-101， HDAC/EGFR/HER2 Inhibitor 
CUDC-101， HDAC/EGFR/HER2 Inhibitor
$69.00 
Catalog No. M60092
A potent multi-target inhibitor targeting HDAC, EGFR and HER2 in clinical trial.
CUDC-907, PI3K/HDAC dual inhibitorCUDC-907, PI3K/HDAC dual inhibitor
CUDC-907, PI3K/HDAC dual inhibitor
$139.00 
Catalog No. M60077
A potent dual inhibitor of class I PI3K kinases and HDACs in clinical trials.
Custom synthesis product 1Custom synthesis product 1
Custom synthesis product 1
$5000.00 
Catalog No. CS-1
CX-4945, CK2 (Casein Kinase 2) InhibitorCX-4945, CK2 (Casein Kinase 2) Inhibitor
CX-4945, CK2 (Casein Kinase 2) Inhibitor
$129.00 
Catalog No. M60267
A potent, selective and bioavailable CK2 (Casein Kinase 2) Inhibitor.
CX-5461, RNA Polymerase I inhibitorCX-5461, RNA Polymerase I inhibitor
CX-5461, RNA Polymerase I inhibitor
$149.00 
Catalog No. M66052
A potent and selective RNA Polymerase I inhibitor, for anti-tumor use.
Cyclopamine, Hedgehog AntagonistCyclopamine, Hedgehog Antagonist
Cyclopamine, Hedgehog Antagonist
$79.00 
Catalog No. M60022
A potent natural product of Hedgehog antagonist; directly binding to the Smoothened/Smo.
Cyclosporin A, MPTP Inhibitor and HSC ProtectorCyclosporin A, MPTP Inhibitor and HSC Protector
Cyclosporin A, MPTP Inhibitor and HSC Protector
$39.00 
Catalog No. M60262
An inhibitor of the mitochondrial permeability transition pore (MPTP).
Daidzein-2c, Osteogenic ModulatorDaidzein-2c, Osteogenic Modulator
Daidzein-2c, Osteogenic Modulator
$109.00 
Catalog No. M60158
A potent synthetic daidzein analog with osteogenic induction potentials on human Mesenchymal Stem Cells (MSC).
Daminozide --- KDM2/7 Histone Demethylases InhibitorDaminozide --- KDM2/7 Histone Demethylases Inhibitor
Daminozide --- KDM2/7 Histone Demethylases Inhibitor
$69.00 
Catalog No. M60074
A potent and selective small molecule inhibitor of the KDM2/7 family of human JmjC histone demethylases.
DAPT, γ-secretase  InhibitorDAPT, γ-secretase  Inhibitor
DAPT, γ-secretase Inhibitor
$300.00 
Catalog No. M60023
A γ-secretase inhibitor and widely used as a Notch pathway inhibitor.
DASA-58 (ML203), Pyruvate Kinase M2 (PKM2) ActivatorDASA-58 (ML203), Pyruvate Kinase M2 (PKM2) Activator
DASA-58 (ML203), Pyruvate Kinase M2 (PKM2) Activator
$109.00 
Catalog No. M60305
A potent and selective Pyruvate kinase M2 (PKM2) activator.
Deltarasin, KRAS-PDEδ InhibitorDeltarasin, KRAS-PDEδ Inhibitor
Deltarasin, KRAS-PDEδ Inhibitor
$139.00 
Catalog No. M60218
A potent and selective small molecular inhibitor of KRAS-PDEδ interaction
demodemo
demo
$0.00 
Catalog No. 123456
DMOG, Prolyl 4-hydroxylase (P4H) InhibitorDMOG, Prolyl 4-hydroxylase (P4H) Inhibitor
DMOG, Prolyl 4-hydroxylase (P4H) Inhibitor
$39.00 
Catalog No. M60287
A selective, competitive and cell permeable prolyl 4-hydroxylase (P4H) inhibitor.
DMXAA (Vadimezan), mSTING AgonistDMXAA (Vadimezan), mSTING Agonist
DMXAA (Vadimezan), mSTING Agonist
$79.00 
Catalog No. M60301
A potent and selective mSTING agonist, selective for mouse STING over human STING.
DNMT3A Polyclonal AntibodyDNMT3A Polyclonal Antibody
DNMT3A Polyclonal Antibody
$0.00 
Catalog No. A70035
DNA (cytosine-5)-methyltransferase 3A (DNMT3A)
DZNep (3-Deazaneplanocin A) --- Histone Methyltransferase Inhibitor DZNep (3-Deazaneplanocin A) --- Histone Methyltransferase Inhibitor 
DZNep (3-Deazaneplanocin A) --- Histone Methyltransferase Inhibitor
$129.00 
Catalog No. M60141
An S-adenosylhomocysteine hydrolase inhibitor, indirectly inhibiting histone methyltransferases and decreasing global DNA methylation
EED226, PRC2 InhibitorEED226, PRC2 Inhibitor
EED226, PRC2 Inhibitor
$139.00 
Catalog No. M60327
A potent and selective allosteric PRC2 inhibitor that directly binds to the H3K27me3 binding pocket of EED.
EML425, CBP/p300 InhibitorEML425, CBP/p300 Inhibitor
EML425, CBP/p300 Inhibitor
$129.00 
Catalog No. M60257
A selective, noncompetitive and cell permeable KAT3 histone acetyltransferases CBP/p300 inhibitor.
Entinostat (MS-275) -- HDAC Inhibitor Entinostat (MS-275) -- HDAC Inhibitor 
Entinostat (MS-275) -- HDAC Inhibitor
$59.00 
Catalog No. M60174
Entinostat (MS-275) is a potent and selective HDAC1 and HDAC3 inhibitor.
EPZ-5676 --- DOT1L inhibitorEPZ-5676 --- DOT1L inhibitor
EPZ-5676 --- DOT1L inhibitor
$139.00 
Catalog No. M60123
A highly potent and selective inhibitor of DOT1L methyltransferase with Ki of 70 pM, selectively blocking the binding of the cofactor, S-adenosylmethionine.
EPZ-6438, EZH2 Methyltransferase InhibitorEPZ-6438, EZH2 Methyltransferase Inhibitor
EPZ-6438, EZH2 Methyltransferase Inhibitor
$129.00 
Catalog No. M60122
EPZ-6438 (E7438) is a potent and selective small molecule inhibitor of histone methyltransferase EZH2 in clinical development.
EPZ015666 (GSK3235025), PRMT5 Inhibitor EPZ015666 (GSK3235025), PRMT5 Inhibitor 
EPZ015666 (GSK3235025), PRMT5 Inhibitor
$129.00 
Catalog No. M60254
A potent, selective and orally bioavailable Protein arginine methyltransferase-5 (PRMT5) Inhibitor.
EX-527, SIRT1 InhibitorEX-527, SIRT1 Inhibitor
EX-527, SIRT1 Inhibitor
$69.00 
Catalog No. M60108
EX-527 is a highly potent and selective inhibitor of SIRT1 with an IC50 ~98 nM.
EZH2 Polyclonal AntibodyEZH2 Polyclonal Antibody
EZH2 Polyclonal Antibody
$0.00 
Catalog No. A70036
Histone-lysine N-methyltransferase EZH2
FASCIN-G2, Fascin InhibitorFASCIN-G2, Fascin Inhibitor
FASCIN-G2, Fascin Inhibitor
$129.00 
Catalog No. M60269
A potent, selective and bioavailable small molecule that inhibits the actin-bundling activity of fascin.
Fatostatin A, Sterol Regulatory Binding Proteins (SREBPs) InhibitorFatostatin A, Sterol Regulatory Binding Proteins (SREBPs) Inhibitor
Fatostatin A, Sterol Regulatory Binding Proteins (SREBPs) Inhibitor
$59.00 
Catalog No. M60180
Fatostatin A is a highly potent, specific and cell permeable inhibitor of Sterol Regulatory Binding Proteins (SREBPs).
Ferrostatin-1 (Fer-1), Ferroptosis Inhibitor Ferrostatin-1 (Fer-1), Ferroptosis Inhibitor 
Ferrostatin-1 (Fer-1), Ferroptosis Inhibitor
$109.00 
Catalog No. M60042
Ferrostatin-1 (Fer-1) is a potent inhibitor of ferroptosis with an EC50 ~60 nM, identified by a HTS using erastin-induced ferroptosis in HT-1080 cells.
FG-4592 (Roxadustat), HIF Prolyl-Hydroxylases InhibitorFG-4592 (Roxadustat), HIF Prolyl-Hydroxylases Inhibitor
FG-4592 (Roxadustat), HIF Prolyl-Hydroxylases Inhibitor
$39.00 
Catalog No. M60263
A potent, selective and bioavailable inhibitor of hypoxia-inducible factor prolyl hydroxylase.
FH1, Hepatocytes Functional EnhancerFH1, Hepatocytes Functional Enhancer
FH1, Hepatocytes Functional Enhancer
$139.00 
Catalog No. M60127
FH1 is a potent and selective small molecule that enhances hepatocyte functions and promotes the differentiation and maturation of iPSC-derived hepatocytes toward a more mature phenotype in vitro.
FLI-06, Notch Pathway ModulatorFLI-06, Notch Pathway Modulator
FLI-06, Notch Pathway Modulator
$139.00 
Catalog No. M60149
FLI-06 is a novel potent and selective small molecule intercepting Notch signaling and the early secretory pathway (EC50 ~2.3 µM), identified by using automated microscopy to monitor the trafficking and processing of a ligand-independent Notch-GFP fusion reporter.
Fmoc-Ala-Ala-Asn-PAB-PNPFmoc-Ala-Ala-Asn-PAB-PNP
Fmoc-Ala-Ala-Asn-PAB-PNP
Inquiry 
Catalog No. L60002
Peptide prodrug linker
Fmoc-Val-Cit-PABFmoc-Val-Cit-PAB
Fmoc-Val-Cit-PAB
Inquiry 
Catalog No. L60001
Peptide prodrug linker
Forskolin, Adenylyl Cyclase Activator Forskolin, Adenylyl Cyclase Activator 
Forskolin, Adenylyl Cyclase Activator
$79.00 
Catalog No. M60024
A potent adenylate cyclase activator to increase the in|tracellular levels of cAMP.
FPH1, Hepatocytes Functional Proliferation InducerFPH1, Hepatocytes Functional Proliferation Inducer
FPH1, Hepatocytes Functional Proliferation Inducer
$139.00 
Catalog No. M60126
FPH1 is a potent and selective small molecule that induced Functional Proliferation of primary human Hepatocytes in vitro, identified by a high-throughput, cell-based screening using primary human hepatocytes.
Furamidine, PRMT1 InhibitorFuramidine, PRMT1 Inhibitor
Furamidine, PRMT1 Inhibitor
$99.00 
Catalog No. M60256
A potent, selective and cell permeable Protein arginine methyltransferase-1 (PRMT1) inhibitor.
GDC-0068, Akt Inhibitor GDC-0068, Akt Inhibitor 
GDC-0068, Akt Inhibitor
$159.00 
Catalog No. M60066
A novel potent and selective ATP competitive Akt inhibitor in clinical trials.
GDC-0349, mTOR Inhibitor GDC-0349, mTOR Inhibitor 
GDC-0349, mTOR Inhibitor
$129.00 
Catalog No. M60110
A potent and selective ATP-competitive inhibitor of mTOR in clinical trials.
GDC-0449 (Vismodegib), Hedgehog Antagonist GDC-0449 (Vismodegib), Hedgehog Antagonist 
GDC-0449 (Vismodegib), Hedgehog Antagonist
$79.00 
Catalog No. M60034
A potent and specific hedgehog pathway inhibitor approved by FDA
GDC-0941,  PI3K Inhibitor GDC-0941,  PI3K Inhibitor 
GDC-0941, PI3K Inhibitor
$79.00 
Catalog No. M60111
A highly potent, selective and orally bioavailable class-I PI3K kinase inhibitor.
GN44028, HIF-1α InhibitorGN44028, HIF-1α Inhibitor
GN44028, HIF-1α Inhibitor
$89.00 
Catalog No. M60325
A potent and selective HIF-1α inhibitor.
GNF-7, Ras Signaling InhibitorGNF-7, Ras Signaling Inhibitor
GNF-7, Ras Signaling Inhibitor
$129.00 
Catalog No. M60281
A potent, selective and bioavailable Ras signaling inhibitor.
GNF4877, β Cell Proliferation Inducer GNF4877, β Cell Proliferation Inducer 
GNF4877, β Cell Proliferation Inducer
$159.00 
Catalog No. M60294
A highly potent and selective small molecule that promotes pancreatic β cell proliferation in rodent and human primary islets.
GNF7156, β Cell Proliferation Inducer GNF7156, β Cell Proliferation Inducer 
GNF7156, β Cell Proliferation Inducer
$139.00 
Catalog No. M60293
A highly potent and selective small molecule that promotes pancreatic β cell proliferation in rodent and human primary islets.
Go6893, PKC InhibitorGo6893, PKC Inhibitor
Go6893, PKC Inhibitor
$129.00 
Catalog No. M60273
A potent pan-PKC inhibitor.
GPR39-C3, GPR39 AgonistGPR39-C3, GPR39 Agonist
GPR39-C3, GPR39 Agonist
$139.00 
Catalog No. M60209
The first potent, selective and orally bioavailable GPR39 agonist.
GPR39-C3bulkGPR39-C3bulk
GPR39-C3bulk
$0.00   $875.00 
Catalog No. M60209-b
GS143, IkappaB Ubiquitination Inhibitor GS143, IkappaB Ubiquitination Inhibitor 
GS143, IkappaB Ubiquitination Inhibitor
$129.00 
Catalog No. M60308
A selective β-TrCP1 ligase inhibitor
GSK-J1, H3K27 Histone Demethylases UTX and JMJD3 Inhibitor GSK-J1, H3K27 Histone Demethylases UTX and JMJD3 Inhibitor 
GSK-J1, H3K27 Histone Demethylases UTX and JMJD3 Inhibitor
$109.00 
Catalog No. M60062
The first selective and potent inhibitor of the H3K27 histone demethylases UTX and JMJD3.
GSK-J4, H3K27 Histone Demethylases UTX and JMJD3 Inhibitor GSK-J4, H3K27 Histone Demethylases UTX and JMJD3 Inhibitor 
GSK-J4, H3K27 Histone Demethylases UTX and JMJD3 Inhibitor
$109.00 
Catalog No. M60063
An ethyl ester derivative of GSK-J1 as a pro-drug for cellular assays; the first selective and potent inhibitor of the H3K27 histone demethylases UTX and JMJD3.
GSK-J4bulkGSK-J4bulk
GSK-J4bulk
$0.00 
Catalog No. M60063-b
GSK-LSD1, LSD1 InhibitorGSK-LSD1, LSD1 Inhibitor
GSK-LSD1, LSD1 Inhibitor
$139.00 
Catalog No. M60179
A highly potent, specific and irreversible inhibitor of Lysine Specific Demethylase-1 (LSD1).
GSK126, EZH2 Methyltransferase Inhibitor.GSK126, EZH2 Methyltransferase Inhibitor.
GSK126, EZH2 Methyltransferase Inhibitor.
$129.00 
Catalog No. M60071
GSK126 is a highly potent and selective small molecule inhibitor of histone methyltransferase EZH2.
GSK126bulkGSK126bulk
GSK126bulk
$0.00 
Catalog No. M60071-b
GSK2801, Bromodomain BAZ2A/B InhibitorGSK2801, Bromodomain BAZ2A/B Inhibitor
GSK2801, Bromodomain BAZ2A/B Inhibitor
$129.00 
Catalog No. M60283
A potent, selective and cell permeable inhibitor of the bromodomain BAZ2A and BAZ2B.
GSK2879552, LSD1 InhibitorGSK2879552, LSD1 Inhibitor
GSK2879552, LSD1 Inhibitor
$129.00 
Catalog No. M60297
A highly potent, selective and orally bioavailable irreversible inhibitor of Lysine Specific Demethylase 1 (LSD1).
GSK343, EZH2 Methyltransferase InhibitorGSK343, EZH2 Methyltransferase Inhibitor
GSK343, EZH2 Methyltransferase Inhibitor
$79.00 
Catalog No. M60173
GSK343 is a potent and selective small molecule inhibitor of histone methyltransferase EZH2.
GSK591 (EPZ015866), PRMT5 InhibitorGSK591 (EPZ015866), PRMT5 Inhibitor
GSK591 (EPZ015866), PRMT5 Inhibitor
$109.00 
Catalog No. M60321
A potent and selective Protein arginine methyltransferase-5 (PRMT5) Inhibitor.
GSK5959, BRPF1 Bromodomain InhibitorGSK5959, BRPF1 Bromodomain Inhibitor
GSK5959, BRPF1 Bromodomain Inhibitor
$129.00 
Catalog No. M60239
A potent, selective and cell permeable BRPF1 bromodomain inhibitor.
H3K36me3 Mouse Monoclonal AntibodyH3K36me3 Mouse Monoclonal Antibody
H3K36me3 Mouse Monoclonal Antibody
$0.00 
Catalog No. A90004
H3K36me3 Mouse Monoclonal Antibody
H3K4me1 Polyclonal AntibodyH3K4me1 Polyclonal Antibody
H3K4me1 Polyclonal Antibody
Inquiry 
Catalog No. A70010
Monomethylated H3K4 Polyclonal Antibody
H3K4me3 Mouse Monoclonal AntibodyH3K4me3 Mouse Monoclonal Antibody
H3K4me3 Mouse Monoclonal Antibody
Inquiry 
Catalog No. A90006
H3K4me3 Mouse Monoclonal Antibody
H3K79me1 Mouse Monoclonal AntibodyH3K79me1 Mouse Monoclonal Antibody
H3K79me1 Mouse Monoclonal Antibody
Inquiry 
Catalog No. A90001
H3K79me1 Mouse Monoclonal Antibody
H3K79me2 Mouse Monoclonal AntibodyH3K79me2 Mouse Monoclonal Antibody
H3K79me2 Mouse Monoclonal Antibody
Inquiry 
Catalog No. A90002
H3K79me2 Mouse Monoclonal Antibody
H3K79me3 Mouse Monoclonal AntibodyH3K79me3 Mouse Monoclonal Antibody
H3K79me3 Mouse Monoclonal Antibody
Inquiry 
Catalog No. A90003
H3K79me3 Mouse Monoclonal Antibody
H3K9(Ac)K14(Ac) Rabbit pAbH3K9(Ac)K14(Ac) Rabbit pAb
H3K9(Ac)K14(Ac) Rabbit pAb
$250.00 
Catalog No. A-10001-100
H3K9me3 Mouse Monoclonal AntibodyH3K9me3 Mouse Monoclonal Antibody
H3K9me3 Mouse Monoclonal Antibody
Inquiry 
Catalog No. A90005
H3K9me3 Mouse Monoclonal Antibody
Harmine, DYRK1A InhibitorHarmine, DYRK1A Inhibitor
Harmine, DYRK1A Inhibitor
$29.00 
Catalog No. M60241
A potent, selective and orally bioavailable DYRK1A inhibitor.
HBX41108, USP7 InhibitorHBX41108, USP7 Inhibitor
HBX41108, USP7 Inhibitor
$129.00 
Catalog No. M60244
A potent and selective ubiquitin-specific protease 7 (USP7) inhibitor.
HCI-2509 (SP2509),  Reversible LSD1 Inhibitor.HCI-2509 (SP2509),  Reversible LSD1 Inhibitor.
HCI-2509 (SP2509), Reversible LSD1 Inhibitor.
$109.00 
Catalog No. M60160
A highly potent, specific, and reversible Lysine Specific Demethylase-1 (LSD1) inhibitor with in vivo efficacy.
HDAC4 Mouse Monoclonal AntibodyHDAC4 Mouse Monoclonal Antibody
HDAC4 Mouse Monoclonal Antibody
Inquiry 
Catalog No. A90011
Histone deacetylase 4 (HDAC4) is a histone deacetylase that represses transcription when tethered to a promoter.
HDAC4 Polyclonal AntibodyHDAC4 Polyclonal Antibody
HDAC4 Polyclonal Antibody
Inquiry 
Catalog No. A70037
Histone deacetylase 4
Heclin, HECT E3 Ubiquitin Ligase InhibitorHeclin, HECT E3 Ubiquitin Ligase Inhibitor
Heclin, HECT E3 Ubiquitin Ligase Inhibitor
$89.00 
Catalog No. M60248
A selective HECT E3 ubiquitin ligase inhibitor to inhibit Nedd4, Smurf2 and WWP1.
HG-10-102-01, LRRK2 Inhibitor HG-10-102-01, LRRK2 Inhibitor 
HG-10-102-01, LRRK2 Inhibitor
$139.00 
Catalog No. M60061
A brain penetrant potent and selective inhibitor of wild-type LRRK2 and the G2019S mutant.
Hh-Ag1.5, Hedgehog Agonist Hh-Ag1.5, Hedgehog Agonist 
Hh-Ag1.5, Hedgehog Agonist
$139.00 
Catalog No. M60004
The most potent and selective agonist of the Hh pathway (Smoothened/Smo agonist); could replace the recombinant Hh protein to activate the Hh pathway
HIF-C2, HIF-2 Inhibitor HIF-C2, HIF-2 Inhibitor 
HIF-C2, HIF-2 Inhibitor
$139.00 
Catalog No. M60121
A potent and selective allosteric inhibitor of hypoxia inducible factor-2 (HIF-2).
Histone H3K27me1 Polyclonal AntibodyHistone H3K27me1 Polyclonal Antibody
Histone H3K27me1 Polyclonal Antibody
Inquiry 
Catalog No. A70013
histone H3 containing the monomethylated lysine 27
Histone H3K27me2 Polyclonal AntibodyHistone H3K27me2 Polyclonal Antibody
Histone H3K27me2 Polyclonal Antibody
Inquiry 
Catalog No. A70014
histone H3 containing the dimethylated lysine 27
Histone H3K27me3 Polyclonal AntibodyHistone H3K27me3 Polyclonal Antibody
Histone H3K27me3 Polyclonal Antibody
Inquiry 
Catalog No. A70015
histone H3 containing the trimethylated lysine 27
Histone H3K36me1 Polyclonal AntibodyHistone H3K36me1 Polyclonal Antibody
Histone H3K36me1 Polyclonal Antibody
Inquiry 
Catalog No. A70016
histone H3 containing the monomethylated lysine 36
Histone H3K36me2 Polyclonal AntibodyHistone H3K36me2 Polyclonal Antibody
Histone H3K36me2 Polyclonal Antibody
Inquiry 
Catalog No. A70017
histone H3 containing the dimethylated lysine 36
Histone H3K36me3 Polyclonal AntibodyHistone H3K36me3 Polyclonal Antibody
Histone H3K36me3 Polyclonal Antibody
Inquiry 
Catalog No. A70018
histone H3 containing the trimethylated lysine 36
Histone H3K4me2 Polyclonal AntibodyHistone H3K4me2 Polyclonal Antibody
Histone H3K4me2 Polyclonal Antibody
Inquiry 
Catalog No. A70011
histone H3 containing the dimethylated lysine 4
Histone H3K4me3 Polyclonal AntibodyHistone H3K4me3 Polyclonal Antibody
Histone H3K4me3 Polyclonal Antibody
Inquiry 
Catalog No. A70012
histone H3 containing the trimethylated lysine 4
Histone H3K79me1 Polyclonal AntibodyHistone H3K79me1 Polyclonal Antibody
Histone H3K79me1 Polyclonal Antibody
Inquiry 
Catalog No. A70019
histone H3 containing the monomethylated lysine 79
Histone H3K79me2 Polyclonal AntibodyHistone H3K79me2 Polyclonal Antibody
Histone H3K79me2 Polyclonal Antibody
Inquiry 
Catalog No. A70020
histone H3 containing the dimethylated lysine 79
Histone H3K79me3 Polyclonal AntibodyHistone H3K79me3 Polyclonal Antibody
Histone H3K79me3 Polyclonal Antibody
Inquiry 
Catalog No. A70021
histone H3 containing the trimethylated lysine 79
Histone H3K9me1 Polyclonal AntibodyHistone H3K9me1 Polyclonal Antibody
Histone H3K9me1 Polyclonal Antibody
Inquiry 
Catalog No. A70022
histone H3 containing the monomethylated lysine 9
Histone H3K9me2 Polyclonal AntibodyHistone H3K9me2 Polyclonal Antibody
Histone H3K9me2 Polyclonal Antibody
Inquiry 
Catalog No. A70023
histone H3 containing the dimethylated lysine 9
Histone H3K9me3 Polyclonal AntibodyHistone H3K9me3 Polyclonal Antibody
Histone H3K9me3 Polyclonal Antibody
Inquiry 
Catalog No. A70024
histone H3 containing the trimethylated lysine 9
Histone H3R26me1 Polyclonal AntibodyHistone H3R26me1 Polyclonal Antibody
Histone H3R26me1 Polyclonal Antibody
Inquiry 
Catalog No. A70031
histone H3 containing the monomethylated Arg26
Histone H3R26me2a Polyclonal AntibodyHistone H3R26me2a Polyclonal Antibody
Histone H3R26me2a Polyclonal Antibody
Inquiry 
Catalog No. A70032
histone H3 containing the asymmetrically dimethylated Arg26
Histone H3R2me1 Polyclonal AntibodyHistone H3R2me1 Polyclonal Antibody
Histone H3R2me1 Polyclonal Antibody
Inquiry 
Catalog No. A70029
histone H3 containing the monomethylated Arg2
Histone H3R2me2a Polyclonal AntibodyHistone H3R2me2a Polyclonal Antibody
Histone H3R2me2a Polyclonal Antibody
Inquiry 
Catalog No. A70028
histone H3 containing the asymmetrically dimethylated Arg2
Histone H3R2me2s Polyclonal AntibodyHistone H3R2me2s Polyclonal Antibody
Histone H3R2me2s Polyclonal Antibody
Inquiry 
Catalog No. A70030
histone H3 containing the symmetrically dimethylated Arg2
Histone H4R3me1 Polyclonal AntibodyHistone H4R3me1 Polyclonal Antibody
Histone H4R3me1 Polyclonal Antibody
Inquiry 
Catalog No. A70025
histone H4 containing the monomethylated Arg3
Histone H4R3me2a Polyclonal AntibodyHistone H4R3me2a Polyclonal Antibody
Histone H4R3me2a Polyclonal Antibody
Inquiry 
Catalog No. A70027
histone H4 containing the asymmetrically dimethylated Arg3
Histone H4R3me2s Polyclonal AntibodyHistone H4R3me2s Polyclonal Antibody
Histone H4R3me2s Polyclonal Antibody
Inquiry 
Catalog No. A70026
histone H4 containing the symmetrically dimethylated Arg3
HLCL-61, PRMT5 InhibitorHLCL-61, PRMT5 Inhibitor
HLCL-61, PRMT5 Inhibitor
$109.00 
Catalog No. M60320
A potent and selective Protein arginine methyltransferase-5 (PRMT5) Inhibitor.
HLY78, Wnt ActivatorHLY78, Wnt Activator
HLY78, Wnt Activator
$149.00 
Catalog No. M60140
An activator of the Wnt pathway by targeting the DIX domain of Axin and potentiating the Axin–LRP6 association, thus promoting LRP6 phosphorylation and Wnt signaling transduction.
HPOB, HDAC6 InhibitorHPOB, HDAC6 Inhibitor
HPOB, HDAC6 Inhibitor
$79.00 
Catalog No. M60231
A potent and selective HDAC6 inhibitor.
Hydroxychloroquine (HCQ), Autophagy and TLR9 Inhibitor Hydroxychloroquine (HCQ), Autophagy and TLR9 Inhibitor 
Hydroxychloroquine (HCQ), Autophagy and TLR9 Inhibitor
$49.00 
Catalog No. M60302
A potent autophagy inhibitor and TLR9 inhibitor
I-BET151 (GSK1210151A), BET Inhibitor I-BET151 (GSK1210151A), BET Inhibitor 
I-BET151 (GSK1210151A), BET Inhibitor
$109.00 
Catalog No. M66053
A potent and selective inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3, and BRD4.
I-BET762  (GSK525762), BET Inhibitor I-BET762  (GSK525762), BET Inhibitor 
I-BET762 (GSK525762), BET Inhibitor
$139.00 
Catalog No. M60154
A novel, highly potent, selective and cell permeable BET inhibitor in clinical trials.
I-BRD9, Bromodomain Containing Protein 9 (BRD9) InhibitorI-BRD9, Bromodomain Containing Protein 9 (BRD9) Inhibitor
I-BRD9, Bromodomain Containing Protein 9 (BRD9) Inhibitor
$129.00 
Catalog No. M60276
A potent, selective and cell permeable Bromodomain Containing Protein 9 (BRD9) inhibitor.
I-CBP112, p300/CBP Bromodomain Inhibitor I-CBP112, p300/CBP Bromodomain Inhibitor 
I-CBP112, p300/CBP Bromodomain Inhibitor
$139.00 
Catalog No. M60128
A highly potent and selective p300/CBP bromodomain inhibitor.
ID-8, DYRK| InhibitorID-8, DYRK| Inhibitor
ID-8, DYRK| Inhibitor
$89.00 
Catalog No. M60102
A potent and selective small molecule inhibitor of dual-specificity tyrosine phosphorylation- regulated kinase (DYRK).
IDH-C227, IDH1 Inhibitor IDH-C227, IDH1 Inhibitor 
IDH-C227, IDH1 Inhibitor
$139.00 
Catalog No. M60043
A potent and selective inhibitor of the IDH1 R132H mutant with good cellular activity.
IDH2-C100, IHD2 Inhibitor IDH2-C100, IHD2 Inhibitor 
IDH2-C100, IHD2 Inhibitor
$129.00 
Catalog No. M60190
A potent and selective inhibitor of IDH2 R140Q and R172K mutant.
IDH2-C100BulkIDH2-C100Bulk
IDH2-C100Bulk
$750.00   $990.00 
Catalog No. M60190-b
iN-LSCiN-LSC
iN-LSC
$89.00 
Catalog No. S10004
Combination of LDN193189 (BMP inhibitor), SB431542 (TGFβ inhibitor), and CHIR99021 (GSK3 inhibitor) can enhance reprogramming of human fibroblasts into induced neurons.
INCB024360 (Epacadostat), IDO InhibitorINCB024360 (Epacadostat), IDO Inhibitor
INCB024360 (Epacadostat), IDO Inhibitor
$109.00 
Catalog No. M60292
A potent and selective indoleamine 2,3-dioxygenase (IDO1) inhibitor.
INDY, DYRK1A/B  InhibitorINDY, DYRK1A/B  Inhibitor
INDY, DYRK1A/B Inhibitor
$79.00 
Catalog No. M60242
A potent and selective DYRK1A/B inhibitor.
IOX1, 2OG Oxygenases InhibitorIOX1, 2OG Oxygenases Inhibitor
IOX1, 2OG Oxygenases Inhibitor
$109.00 
Catalog No. M60195
A cell-permeable broad-spectrum inhibitor of most 2OG oxygenases.
IOX2, HIF Prolyl-Hydroxylases (PHD2) Inhibitor IOX2, HIF Prolyl-Hydroxylases (PHD2) Inhibitor 
IOX2, HIF Prolyl-Hydroxylases (PHD2) Inhibitor
$89.00 
Catalog No. M66054
A potent and selective PHD (HIF prolyl-hydroxylases) inhibitor with cellular activity.
IOX4, PHD2 InhibitorIOX4, PHD2 Inhibitor
IOX4, PHD2 Inhibitor
$109.00 
Catalog No. M60284
A potent and selective PHD2 inhibitor.
iPSC-TSPCiPSC-TSPC
iPSC-TSPC
$109.00 
Catalog No. S10005
Combination of Thiazovivin (ROCK inhibitor), SB431542 (TGFβ inhibitor), PD0325901 (MEK inhibitor), and CHIR99021 (GSK3 inhibitor) can enhance and accelerate reprogramming of human somatic cells (e.g., fibroblasts) into iPSCs.
IRE-3, IRE1a Modulator IRE-3, IRE1a Modulator 
IRE-3, IRE1a Modulator
$129.00 
Catalog No. M60167
A highly potent and selective small molecule modulator of IRE1α.
Ischemin, CBP Bromodomain Inhibitor Ischemin, CBP Bromodomain Inhibitor 
Ischemin, CBP Bromodomain Inhibitor
$79.00 
Catalog No. M60229
A potent, selective and cell permeable CBP bromodomain inhibitor.
ISRIB (trans-isomer), Inhibitor of “Integrated Stress Response” (ISR)ISRIB (trans-isomer), Inhibitor of “Integrated Stress Response” (ISR)
ISRIB (trans-isomer), Inhibitor of “Integrated Stress Response” (ISR)
$129.00 
Catalog No. M60125
A potent and selective small molecule inhibitor of PERK signaling that can potently reverse the effects of eIF2α phosphorylation, Inhibitor of “Integrated Stress Response” (ISR).
ISX9, Neurogenic ModulatorISX9, Neurogenic Modulator
ISX9, Neurogenic Modulator
$99.00 
Catalog No. M60274
A neurogenic modulator.
ITD-1, TGFβ inhibitor ITD-1, TGFβ inhibitor 
ITD-1, TGFβ inhibitor
$139.00 
Catalog No. M60060
A highly selective TGFβ inhibitor promotes cardiomyogenesis in embryonic stem cells.
IU1, Proteasome USP14  Inhibitor IU1, Proteasome USP14  Inhibitor 
IU1, Proteasome USP14 Inhibitor
$49.00 
Catalog No. M60203
A cell-permeable, reversible and selective inhibitor of human proteasome USP14.
IWP-2, Porcupine (Wnt) Inhibitor IWP-2, Porcupine (Wnt) Inhibitor 
IWP-2, Porcupine (Wnt) Inhibitor
$79.00 
Catalog No. M60115
A potent and highly selective Wnt signaling antagonist targeting porcupine.
J147, Neuroprotective Small MoleculeJ147, Neuroprotective Small Molecule
J147, Neuroprotective Small Molecule
$89.00 
Catalog No. M60012
A potent and orally active neurotrophic molecule with broadly neuroprotective efficacy in vitro and in vivo.
JIB-04 (NSC693627), Jumonji Histone Demethylase InhibitorJIB-04 (NSC693627), Jumonji Histone Demethylase Inhibitor
JIB-04 (NSC693627), Jumonji Histone Demethylase Inhibitor
$119.00 
Catalog No. M60132
A potent, selective and cell permeable Jumonji histone demethylase inhibitor, not a competitive inhibitor of a-ketoglutarate.
JK184, Hedgehog Antagonist JK184, Hedgehog Antagonist 
JK184, Hedgehog Antagonist
$79.00 
Catalog No. M60087
A potent and cell-permeable inhibitor of hedgehog (Hh) signaling downstream of Smo.
JNJ-42041935, HIF-PHD InhibitorJNJ-42041935, HIF-PHD Inhibitor
JNJ-42041935, HIF-PHD Inhibitor
$129.00 
Catalog No. M60285
A potent and selective HIF-PHD inhibitor.
Kartogenin (KGN), Chondrogenesis Modulator Kartogenin (KGN), Chondrogenesis Modulator 
Kartogenin (KGN), Chondrogenesis Modulator
$79.00 
Catalog No. M60027
Selectively promote chondrocyte differentiation of human mesenchymal stem cells.
KDM5 C70bulkKDM5 C70bulk
KDM5 C70bulk
$0.00 
Catalog No. M60192-b
KDM5-C49, JARID1 Histone Demethylases Inhibitor KDM5-C49, JARID1 Histone Demethylases Inhibitor 
KDM5-C49, JARID1 Histone Demethylases Inhibitor
$139.00 
Catalog No. M60191
A potent and selective inhibitor of Jumonji AT-Rich Interactive Domain 1 (JARID1) histone demethylases
KDM5-C49bulkKDM5-C49bulk
KDM5-C49bulk
$0.00 
Catalog No. M60191-b
KDM5-C70, JARID1 Histone Demethylases Inhibitor KDM5-C70, JARID1 Histone Demethylases Inhibitor 
KDM5-C70, JARID1 Histone Demethylases Inhibitor
$139.00 
Catalog No. M60192
An ethyl ester derivative of KDM5-C49, which is a potent and selective inhibitor of Jumonji AT-Rich Interactive Domain 1 (JARID1) histone demethylases.
KL001, Cryptochrome ActivatorKL001, Cryptochrome Activator
KL001, Cryptochrome Activator
$79.00 
Catalog No. M66044
A novel small molecule specifically interacting with cryptochrome (CRY) and causing lengthening of the circadian period.
KRAS-C9, K-Ras(G12C) Inhibitor KRAS-C9, K-Ras(G12C) Inhibitor 
KRAS-C9, K-Ras(G12C) Inhibitor
$139.00 
Catalog No. M60219
A potent and selective allosteric inhibitor of oncogenic K-Ras(G12C).
KY02111, Wnt Inhibitor KY02111, Wnt Inhibitor 
KY02111, Wnt Inhibitor
$109.00 
Catalog No. M60073
A potent and selective Wnt inhibitor promotes differentiation of hESCs/iPSCs to cardiomyocytes; might function downstream from GSK3β and APC in b-catenin destruction complex
KYA1797K, Wnt/β-catenin InhibitorKYA1797K, Wnt/β-catenin Inhibitor
KYA1797K, Wnt/β-catenin Inhibitor
$129.00 
Catalog No. M60317
A highly potent and selective Wnt/β-catenin inhibitor binding directly to the regulators of G-protein signaling domain of axin.
L002 (NSC764414), p300 Inhibitor L002 (NSC764414), p300 Inhibitor 
L002 (NSC764414), p300 Inhibitor
$99.00 
Catalog No. M60198
A novel selective, cell permeable and reversible inhibitor of p300 histone acetyl transferase.
L755,507, CRISPR Editing EnhancerL755,507, CRISPR Editing Enhancer
L755,507, CRISPR Editing Enhancer
$89.00 
Catalog No. M60237
CRISPR editing enhancer to enhance CRISPR-mediated homology-directed repair (HDR) efficiency in human induced pluripotent stem cells (iPSCs) and other cell types.
LDE225, Hedgehog Antagonist LDE225, Hedgehog Antagonist 
LDE225, Hedgehog Antagonist
$99.00 
Catalog No. M60013
A potent and specific Hedgehog pathway inhibitor (Smo antagonist) in clinical trials.
LDN-193189, BMP inhibitor LDN-193189, BMP inhibitor 
LDN-193189, BMP inhibitor
$79.00 
Catalog No. M60008
A highly potent and selective BMP pathway inhibitor (selective for ALK2 and ALK3); can replace Noggin protein in cellular and in vivo use.
LDN-57444, Ubiquitin C-terminal Hydrolase-L1 (UCH-L1) InhibitorLDN-57444, Ubiquitin C-terminal Hydrolase-L1 (UCH-L1) Inhibitor
LDN-57444, Ubiquitin C-terminal Hydrolase-L1 (UCH-L1) Inhibitor
$69.00 
Catalog No. M60204
A novel potent and selective inhibitor of ubiquitin C-terminal hydrolase-L1 (UCH-L1).
LGK974, Porcupine (Wnt) Inhibitor LGK974, Porcupine (Wnt) Inhibitor 
LGK974, Porcupine (Wnt) Inhibitor
$139.00 
Catalog No. M60106
A highly potent, selective and orally bioavailable Porcupine inhibitor (Wnt signaling antagonist) in clinical trials.
Library of Epigenetic compoundsLibrary of Epigenetic compounds
Library of Epigenetic compounds
$7000.00 
Catalog No. LI30001-2
Compound Library of Epigenetic Set is composed of 117 small molecules in separated vials.
LLY-507, Protein-lysine Methyltransferase SMYD2 InhibitorLLY-507, Protein-lysine Methyltransferase SMYD2 Inhibitor
LLY-507, Protein-lysine Methyltransferase SMYD2 Inhibitor
$129.00 
Catalog No. M60259
A potent, selective and cell permeable protein lysine methyltransferase SMYD2 inhibitor.
LMK235, HDAC4 and HDAC5 Inhibitor LMK235, HDAC4 and HDAC5 Inhibitor 
LMK235, HDAC4 and HDAC5 Inhibitor
$89.00 
Catalog No. M60145
A potent and selective histone deacetylase HDAC4 and HDAC5 inhibitor.
LSD1-C76, LSD1 Inhibitor LSD1-C76, LSD1 Inhibitor 
LSD1-C76, LSD1 Inhibitor
$159.00 
Catalog No. M66045
The most potent and selective Lysine Specific Demethylase-1 (LSD1) inhibitor so far.
LY2109761, TGFβ InhibitorLY2109761, TGFβ Inhibitor
LY2109761, TGFβ Inhibitor
$109.00 
Catalog No. M60035
A novel potent and selective TGFβ receptor type I and type II (TβRI/II) dual inhibitor with Ki of 38 nM and 300 nM respectively.
LY2157299, TGFβ Inhibitor LY2157299, TGFβ Inhibitor 
LY2157299, TGFβ Inhibitor
$169.00 
Catalog No. M60064
A novel potent and selective TGFβ receptor type I and type II (TβRI/II) inhibitor with IC50 of 86 nM and 2 nM respectively.
LY2784544, JAK2 inhibitorLY2784544, JAK2 inhibitor
LY2784544, JAK2 inhibitor
$129.00 
Catalog No. M60079
A highly potent and selective mutant JAK2 (V617F) inhibitor.
LY294002, PI3K/BET Dual Inhibitor LY294002, PI3K/BET Dual Inhibitor 
LY294002, PI3K/BET Dual Inhibitor
$79.00 
Catalog No. M60157
A potent and selective small molecule PI3K and BET bromodomain dual inhibitor.
LY411575, γ-secretase Inhibitor LY411575, γ-secretase Inhibitor 
LY411575, γ-secretase Inhibitor
$119.00 
Catalog No. M60078
A highly potent, selective, and orally bioavailable inhibitor of gamma secretase.
MAL-di-EG-OSuMAL-di-EG-OSu
MAL-di-EG-OSu
$0.00 
Catalog No. L600010
Thiol reactive linker
MAL-HA-OSuMAL-HA-OSu
MAL-HA-OSu
Inquiry 
Catalog No. L60005
Thiol reactive linker
MALT1-MI-2 (MI-2), MALT1 inhibitor MALT1-MI-2 (MI-2), MALT1 inhibitor 
MALT1-MI-2 (MI-2), MALT1 inhibitor
$129.00 
Catalog No. M60098
A highly potent and selective small molecule directly binding to MALT1 and irreversibly suppressing its protease function.
MC1568, Class IIa HDAC InhibitorMC1568, Class IIa HDAC Inhibitor
MC1568, Class IIa HDAC Inhibitor
$79.00 
Catalog No. M60224
A potent and selective inhibitor of class IIa histone deacetylases (HDACs), more selective for HD1-A than HD1-B.
ME0328, PARP-3 InhibitorME0328, PARP-3 Inhibitor
ME0328, PARP-3 Inhibitor
$109.00 
Catalog No. M60329
A potent, selective and cell permeable PARP-3 inhibitor.
MEK162 (ARRY-162), MEK InhibitorMEK162 (ARRY-162), MEK Inhibitor
MEK162 (ARRY-162), MEK Inhibitor
$119.00 
Catalog No. M60080
A highly potent, selective, and orally bioavailable MEK inhibitor in clinical trials.
Methoxy-X04, Fluorescent Amyloid β (Aβ) ProbeMethoxy-X04, Fluorescent Amyloid β (Aβ) Probe
Methoxy-X04, Fluorescent Amyloid β (Aβ) Probe
$79.00 
Catalog No. M60135
A fluorescent amyloid β (Aβ) probe for the detection and quantification of plaques, tangles and cerebrovascular amyloid with good specificity.
MHY1485, mTOR ActivatorMHY1485, mTOR Activator
MHY1485, mTOR Activator
$49.00 
Catalog No. M60189
A novel potent, selective and cell-permeable mTOR activator.
MI-2, Menin-MLL Inhibitor MI-2, Menin-MLL Inhibitor 
MI-2, Menin-MLL Inhibitor
$119.00 
Catalog No. M66046
A highly potent and selective small molecule directly binding to MALT1 and irreversibly suppressing its protease function.
MK-1775 (AZD1775), WEE1 Inhibitor MK-1775 (AZD1775), WEE1 Inhibitor 
MK-1775 (AZD1775), WEE1 Inhibitor
$129.00 
Catalog No. M60299
A highly potent, selective and orally bioavailable Wee1 kinase inhibitor.
ML141, Cdc42 GTPase InhibitorML141, Cdc42 GTPase Inhibitor
ML141, Cdc42 GTPase Inhibitor
$109.00 
Catalog No. M60134
A potent, selective and reversible non-competitive inhibitor of Cdc42 GTPase.
ML228, HIF Pathway ActivatorML228, HIF Pathway Activator
ML228, HIF Pathway Activator
$129.00 
Catalog No. M60130
A potent and selective hypoxia inducible factor (HIF) pathway activator.
ML239, Breast Cancer Stem Cell InhibitorML239, Breast Cancer Stem Cell Inhibitor
ML239, Breast Cancer Stem Cell Inhibitor
$129.00 
Catalog No. M60282
A potent and selective breast cancer stem cell inhibitor.
ML323, USP1-UAF1 Inhibitor ML323, USP1-UAF1 Inhibitor 
ML323, USP1-UAF1 Inhibitor
$139.00 
Catalog No. M60188
A potent, selective and reversible inhibitor of the USP1-UAF1 deubiquitinase complex.
ML324, JMJD2 Histone Demethylase Inhibitor ML324, JMJD2 Histone Demethylase Inhibitor 
ML324, JMJD2 Histone Demethylase Inhibitor
$139.00 
Catalog No. M60183
A potent, selective and cell permeable inhibitor of Jumonji domain-containing protein 2 (JMJD2) histone demethylase.
MLN8237 (Alisertib), Aurora A inhibitor MLN8237 (Alisertib), Aurora A inhibitor 
MLN8237 (Alisertib), Aurora A inhibitor
$119.00 
Catalog No. M60093
A highly potent and selective Aurora A inhibitor with >200-fold selective towards Aurora B.
MM-102, WDR5-MLL1 AntagonistMM-102, WDR5-MLL1 Antagonist
MM-102, WDR5-MLL1 Antagonist
$129.00 
Catalog No. M60166
A highly potent and selective inhibitor of the MLL1/WDR5 interaction.
MRT68921, Autophagy Kinase ULK1/2 Inhibitor MRT68921, Autophagy Kinase ULK1/2 Inhibitor 
MRT68921, Autophagy Kinase ULK1/2 Inhibitor
$109.00 
Catalog No. M60311
A potent, selective and dual autophagy kinase ULK1/2 inhibitor.
MS023, PRMT Inhibitor MS023, PRMT Inhibitor 
MS023, PRMT Inhibitor
$109.00 
Catalog No. M60314
A potent, selective and cell permeable type I PRMT inhibitor.
MS049, PRMT4 and PRMT6 Inhibitor MS049, PRMT4 and PRMT6 Inhibitor 
MS049, PRMT4 and PRMT6 Inhibitor
$89.00 
Catalog No. M60310
A potent, selective and cell permeable PRMT4 and PRMT6 inhibitor.
MS436, BRD4 Inhibitor MS436, BRD4 Inhibitor 
MS436, BRD4 Inhibitor
$109.00 
Catalog No. M60232
A potent and selective BET bromodomain inhibitor for BRD4 (1) and BRD4 (2).
MSAB, β-catenin InhibitorMSAB, β-catenin Inhibitor
MSAB, β-catenin Inhibitor
$129.00 
Catalog No. M60316
A potent and selective Wnt/β-catenin inhibitor identified using cell-based chemical screening.
N106, SERCA2a SUMOylation ActivatorN106, SERCA2a SUMOylation Activator
N106, SERCA2a SUMOylation Activator
$129.00 
Catalog No. M60271
A potent SERCA2a SUMOylation activator, which increases SUMOylation of SERCA2a.
N3-tri-EG-OSuN3-tri-EG-OSu
N3-tri-EG-OSu
Inquiry 
Catalog No. L60004
Click chemistry linker
NAB2, Rsp5/Nedd4 pathway activator, rescuing α-synuclein toxicityNAB2, Rsp5/Nedd4 pathway activator, rescuing α-synuclein toxicity
NAB2, Rsp5/Nedd4 pathway activator, rescuing α-synuclein toxicity
$129.00 
Catalog No. M60153
A novel and highly potent small molecule Rsp5/Nedd4 pathway activator that was shown to strongly and selectively protect diverse cell types from α-synuclein toxicity.
Napabucasin (BBI608), STAT3 InhibitorNapabucasin (BBI608), STAT3 Inhibitor
Napabucasin (BBI608), STAT3 Inhibitor
$89.00 
Catalog No. M60303
A potent and selective STAT3 inhibitor.
Neural-LSBNeural-LSB
Neural-LSB
$79.00 
Catalog No. S10001
Combination of LDN193189 (BMP inhibitor) and SB431542 (TGFβ inhibitor) can rapidly and efficiently induce neural differentiation of human ESC and iPSC in 5 days.
Neuronal-LSB3iNeuronal-LSB3i
Neuronal-LSB3i
$329.00 
Catalog No. S10002
Combination of LSB and three other inhibitors/3i (i.e., CHIR99021/GSK3 inhibitor, SU5402/FGF-VEGF-PDGF inhibitor, DAPT/Notch inhibitor) can induce very rapid and efficient neuronal differentiation of human ESC and iPSC into nociceptors.
NI-57, BRPF Bromodomain InhibitorNI-57, BRPF Bromodomain Inhibitor
NI-57, BRPF Bromodomain Inhibitor
$109.00 
Catalog No. M60279
A potent and selective inhibitor of the bromodomain of the BRPFs.
NLG919 (RG6078), IDO InhibitorNLG919 (RG6078), IDO Inhibitor
NLG919 (RG6078), IDO Inhibitor
$129.00 
Catalog No. M60258
A potent, selective and orally bioavailable IDO (indoleamine-(2,3)-dioxygenase) pathway inhibitor.
NMS-859, ATPase VCP/p97 InhibitorNMS-859, ATPase VCP/p97 Inhibitor
NMS-859, ATPase VCP/p97 Inhibitor
$139.00 
Catalog No. M60148
A potent and specific small molecule covalent inhibitor of the ATPase VCP/p97.
NMS-873, ATPase VCP/p97 Inhibitor NMS-873, ATPase VCP/p97 Inhibitor 
NMS-873, ATPase VCP/p97 Inhibitor
$139.00 
Catalog No. M60165
A potent and specific small molecule allosteric inhibitor of the ATPase VCP/p97.
NMS-873/BulkNMS-873/Bulk
NMS-873/Bulk
$0.00 
Catalog No. M60165-b
NSC319726, Mutant p53 Activator NSC319726, Mutant p53 Activator 
NSC319726, Mutant p53 Activator
$89.00 
Catalog No. M66047
A potent and selective activator of the most common p53R175 mutant, restoring the mutant p53 to its WT structure and function.
NSC636819, KDM4A/KDM4B InhibitorNSC636819, KDM4A/KDM4B Inhibitor
NSC636819, KDM4A/KDM4B Inhibitor
$109.00 
Catalog No. M60290
A cell permeable and selective novel active-site KDM4A/KDM4B inhibitor.
NSC697923, Ub-conjugating Enzyme (E2) InhibitorNSC697923, Ub-conjugating Enzyme (E2) Inhibitor
NSC697923, Ub-conjugating Enzyme (E2) Inhibitor
$69.00 
Catalog No. M60202
A cell permeable, potent and selective inhibitor of the Ub-conjugating enzyme (E2) complex Ubc13-Uev1A.
NU9056--- KAT5 (Tip60) Histone Acetyltransferase InhibitorNU9056--- KAT5 (Tip60) Histone Acetyltransferase Inhibitor
NU9056--- KAT5 (Tip60) Histone Acetyltransferase Inhibitor
$69.00 
Catalog No. M60147
A potent and selective KAT5 (Tip60) histone acetyltransferase inhibitor.
NVP-BGT226, PI3K/mTOR Dual InhibitorNVP-BGT226, PI3K/mTOR Dual Inhibitor
NVP-BGT226, PI3K/mTOR Dual Inhibitor
$89.00 
Catalog No. M66050
A PI3K/mTOR dual inhibitor in clinical trials for advanced solid tumors.
NVP-BKM120, PI3K Inhibitor BKM120NVP-BKM120, PI3K Inhibitor BKM120
NVP-BKM120, PI3K Inhibitor BKM120
$89.00 
Catalog No. M66051
A selective PI3K Inhibitor in clinical trials for advanced solid tumors.
NVP-TNKS656, Wnt / Tankyrase Inhibitor NVP-TNKS656, Wnt / Tankyrase Inhibitor 
NVP-TNKS656, Wnt / Tankyrase Inhibitor
$109.00 
Catalog No. M60328
A highly potent, selective and oral bioavailable tankyrase inhibitor for TNKS2.
NVS-SM1, SMN2 Splicing ModulatorNVS-SM1, SMN2 Splicing Modulator
NVS-SM1, SMN2 Splicing Modulator
$129.00 
Catalog No. M60277
A highly potent, selective and orally active small molecule SMN2 splicing modulator enhancing SMN exon 7 inclusion.
NVS-SM1BulkNVS-SM1Bulk
NVS-SM1Bulk
$0.00 
Catalog No. M60277-b
OAC1, Oct4 ActivatorOAC1, Oct4 Activator
OAC1, Oct4 Activator
$109.00 
Catalog No. M60086
A potent Oct4 activator significantly enhancing iPSC reprogramming efficiency and accelerating the reprogramming process.
OF-1, BRPF Bromodomain Inhibitor OF-1, BRPF Bromodomain Inhibitor 
OF-1, BRPF Bromodomain Inhibitor
$129.00 
Catalog No. M60222
A potent and selective BRPF (BRomodomain and PHD Finger containing) inhibitor.
OG-L002, LSD1 InhibitorOG-L002, LSD1 Inhibitor
OG-L002, LSD1 Inhibitor
$89.00 
Catalog No. M60161
A highly potent and specific inhibitor of Lysine Specific Demethylase-1 (LSD1).
OICR9429, WDR5 AntagonistOICR9429, WDR5 Antagonist
OICR9429, WDR5 Antagonist
$129.00 
Catalog No. M60255  
A potent and selective WD repeat-containing protein 5 (WDR5) antagonist.
ONX-0914, Immunoproteasome InhibitorONX-0914, Immunoproteasome Inhibitor
ONX-0914, Immunoproteasome Inhibitor
$139.00 
Catalog No. M60112
A potent and selective immunoproteasome inhibitor.
Optovin, TRPA1 ActivatorOptovin, TRPA1 Activator
Optovin, TRPA1 Activator
$129.00 
Catalog No. M60103
A potent and selective small molecule activator of human| TRPA1.
ORY-1001 (RG-6016), LSD1 InhibitorORY-1001 (RG-6016), LSD1 Inhibitor
ORY-1001 (RG-6016), LSD1 Inhibitor
$129.00 
Catalog No. M60295
A highly potent and selective inhibitor of Lysine Specific Demethylase 1 (LSD1) in phase I/II.
OSI-027, mTOR InhibitorOSI-027, mTOR Inhibitor
OSI-027, mTOR Inhibitor
$109.00 
Catalog No. M60113
OSI-027 is a selective and potent dual inhibitor of mTORC1 and mTORC2
OTX015, BET Inhibitor OTX015, BET Inhibitor 
OTX015, BET Inhibitor
$89.00 
Catalog No. M60193
OTX015 is a novel, highly potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2, BRD3 and BRD4 with IC50 of 10-19 nM.
P22077, USP7 inhibitorP22077, USP7 inhibitor
P22077, USP7 inhibitor
$99.00 
Catalog No. M60019
A potent and selective USP7 inhibitor.
P5091, Ubiquitin-specific Protease 7 (USP7) InhibitorP5091, Ubiquitin-specific Protease 7 (USP7) Inhibitor
P5091, Ubiquitin-specific Protease 7 (USP7) Inhibitor
$79.00 
Catalog No. M60205
P5091 (P005091) is a novel potent and selective inhibitor of ubiquitin-specific protease 7 (USP7)
P7C3, Neuroprotective Small MoleculeP7C3, Neuroprotective Small Molecule
P7C3, Neuroprotective Small Molecule
$119.00 
Catalog No. M60017
A neuroprotective small molecule with favorable in vivo PK; protects newborn neurons from apoptosis.
PBIT, JARID1 Histone Demethylases InhibitorPBIT, JARID1 Histone Demethylases Inhibitor
PBIT, JARID1 Histone Demethylases Inhibitor
$129.00 
Catalog No. M60170
PBIT is a potent, specific, reversible and cell-permeable inhibitor of Jumonji AT-Rich Interactive Domain 1 (JARID1) histone demethylases.
PCI-34051, HDAC8 InhibitorPCI-34051, HDAC8 Inhibitor
PCI-34051, HDAC8 Inhibitor
$79.00 
Catalog No. M60178
PCI-34051 is a potent and selective inhibitor of histone deacetylase 8 (HDAC8).
PD-1/PD-L1 Inhibitor C1PD-1/PD-L1 Inhibitor C1
PD-1/PD-L1 Inhibitor C1
$109.00 
Catalog No. M60312
A potent and selective small molecule inhibitor of the PD-1/PD-L1 protein/protein interactions.
PD0325901, MEK InhibitorPD0325901, MEK Inhibitor
PD0325901, MEK Inhibitor
$69.00 
Catalog No. M60018
A potent and selective MEK inhibitor.
PF-04979064, PI3K/mTOR Dual InhibitorPF-04979064, PI3K/mTOR Dual Inhibitor
PF-04979064, PI3K/mTOR Dual Inhibitor
$149.00 
Catalog No. M60114
PF-04979064 is a highly potent and orally bioavailable PI3K/mTOR dual inhibitor developed through structure-based drug design.
PF-CBP1，CBP/p300 Bromodomain Inhibitor PF-CBP1，CBP/p300 Bromodomain Inhibitor 
PF-CBP1，CBP/p300 Bromodomain Inhibitor
$129.00 
Catalog No. M60313
A potent and selective CBP/p300 bromodomain inhibitor.
PFI-1, BET InhibitorPFI-1, BET Inhibitor
PFI-1, BET Inhibitor
$129.00 
Catalog No. M60120
PFI-1 is a novel potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family proteins BRD2 and BRD4.
PFI-2, SETD7 Histone Lysine Methyltransferase Inhibitor PFI-2, SETD7 Histone Lysine Methyltransferase Inhibitor 
PFI-2, SETD7 Histone Lysine Methyltransferase Inhibitor
$139.00 
Catalog No. M60182
PFI-2 is a novel potent and selective SETD7 histone lysine methyltransferase inhibitor.
PFI-3, SMARCA Bromodomains InhibitorPFI-3, SMARCA Bromodomains Inhibitor
PFI-3, SMARCA Bromodomains Inhibitor
$139.00 
Catalog No. M60175
PFI-3 is a novel potent, selective and cell permeable inhibitor of SMARCA4 and PB1(5) bromodomains.
PFI-4, BRPF1 Bromodomain InhibitorPFI-4, BRPF1 Bromodomain Inhibitor
PFI-4, BRPF1 Bromodomain Inhibitor
$129.00 
Catalog No. M60264
A potent, selective and cell permeable BRPF1 bromodomain inhibitor.
Phospho-HDAC4 (Ser632) AntibodyPhospho-HDAC4 (Ser632) Antibody
Phospho-HDAC4 (Ser632) Antibody
$0.00 
Catalog No. A90009-5
a
Phospho-HDAC4 (Ser632) AntibodyPhospho-HDAC4 (Ser632) Antibody
Phospho-HDAC4 (Ser632) Antibody
$0.00 
Catalog No. A90009
Phospho-HDAC4 (Ser632) Antibody. Histone deacetylase 4 (HDAC4) is a histone deacetylase that represses transcription when tethered to a promoter.
PluriSIn#1, Pluripotent Cell-specific Inhibitor PluriSIn#1, Pluripotent Cell-specific Inhibitor 
PluriSIn#1, Pluripotent Cell-specific Inhibitor
$109.00 
Catalog No. M60085
A potent small molecule to selectively eliminate human pluripotent stem cells/hPSCs while sparing a large array of tissue-specific stem/progenitor and differentiated cells.
pNSC-CSBpNSC-CSB
pNSC-CSB
$69.00 
Catalog No. S10003
Combination of CHIR99021 (GSK3 inhibitor) and SB431542 (TGFβ inhibitor) with human LIF can efficiently induce and long-term homogenously expand primitive neural stem cells from human ESC and iPSC.
PP242, mTORC1/mTORC2 inhibitorPP242, mTORC1/mTORC2 inhibitor
PP242, mTORC1/mTORC2 inhibitor
$69.00 
Catalog No. M60094
A highly potent, selective and ATP-competitive mTORC1/mTORC2 inhibitor.
PR-619, Deubiquitinylating Enzyme (DUB) Inhibitor PR-619, Deubiquitinylating Enzyme (DUB) Inhibitor 
PR-619, Deubiquitinylating Enzyme (DUB) Inhibitor
$59.00 
Catalog No. M60199
PR-619 is a cell-permeable, non-selective, reversible broad-range inhibitor of the deubiquitinylating enzymes (DUBs).
PRMT1-2e, Protein Arginine Methyltransferase 1 (PRMT1) Inhibitor PRMT1-2e, Protein Arginine Methyltransferase 1 (PRMT1) Inhibitor 
PRMT1-2e, Protein Arginine Methyltransferase 1 (PRMT1) Inhibitor
$69.00 
Catalog No. M60181
PRMT1-2e is a potent, specific and cell permeable inhibitor of protein arginine methyltransferase 1 (PRMT1).
PRT4165, E3 Ubiquitin-ligase Bmi1/Ring1A InhibitorPRT4165, E3 Ubiquitin-ligase Bmi1/Ring1A Inhibitor
PRT4165, E3 Ubiquitin-ligase Bmi1/Ring1A Inhibitor
$39.00 
Catalog No. M60245
A potent and selective E3 Ubiquitin-ligase Bmi1/Ring1A Inhibitor.
PS48---PDK1 ActivatorPS48---PDK1 Activator
PS48---PDK1 Activator
$79.00 
Catalog No. M60026
An allosteric small molecule activator of PDK1.
PTC-209, BMI-1 InhibitorPTC-209, BMI-1 Inhibitor
PTC-209, BMI-1 Inhibitor
$129.00 
Catalog No. M60159
PTC-209 is a novel potent and selective BMI-1 inhibitor, targeting the BMI-1 self-renewal machinery.
PTC-209BulkPTC-209Bulk
PTC-209Bulk
$0.00 
Catalog No. M60159-b
Purmorphamine, Hedgehog Agonist Purmorphamine, Hedgehog Agonist 
Purmorphamine, Hedgehog Agonist
$99.00 
Catalog No. M66055
A selective hedgehog pathway agonist (Smo agonist).
PX-478, Hypoxia-inducible Factor-1α (HIF-1α) Inhibitor PX-478, Hypoxia-inducible Factor-1α (HIF-1α) Inhibitor 
PX-478, Hypoxia-inducible Factor-1α (HIF-1α) Inhibitor
$129.00 
Catalog No. M60227
A highly potent and selective Hypoxia-inducible Factor-1α (HIF-1α) inhibitor.
Py-ds-But-OSuPy-ds-But-OSu
Py-ds-But-OSu
Inquiry 
Catalog No. L60003
Disulfide prodrug linker
PYR-41---Ubiquitin-activating Enzyme E1  Inhibitor PYR-41---Ubiquitin-activating Enzyme E1  Inhibitor 
PYR-41---Ubiquitin-activating Enzyme E1 Inhibitor
$59.00 
Catalog No. M60201
PYR-41 is a specific and cell permeable inhibitor of ubiquitin-activating enzyme E1
Pyrintegrin---Cell Survival EnhancerPyrintegrin---Cell Survival Enhancer
Pyrintegrin---Cell Survival Enhancer
$109.00 
Catalog No. M60028
A potent small molecule promoting hESC survival
PYZD-4409, Ubiquitin-activating Enzyme (E1) Inhibitor PYZD-4409, Ubiquitin-activating Enzyme (E1) Inhibitor 
PYZD-4409, Ubiquitin-activating Enzyme (E1) Inhibitor
$139.00 
Catalog No. M60213
A novel potent, selective and cell permeable inhibitor of ubiquitin-activating enzyme (E1).
RA190, Ubiquitin Receptor RPN13/ADRM1 InhibitorRA190, Ubiquitin Receptor RPN13/ADRM1 Inhibitor
RA190, Ubiquitin Receptor RPN13/ADRM1 Inhibitor
$139.00 
Catalog No. M60163
A novel potent and selective inhibitor of proteasome Ubiquitin receptor RPN13/ADRM1.
RA190bulkRA190bulk
RA190bulk
$0.00 
Catalog No. M60163-b
Rapamycin, mTOR inhibitor Rapamycin, mTOR inhibitor 
Rapamycin, mTOR inhibitor
$89.00 
Catalog No. M60029
A potent and selective mTOR inhibitor, directly binding to the mTOR Complex 1 (mTORC1).
Recombinant Human Activin ARecombinant Human Activin A
Recombinant Human Activin A
$3900.00 
Catalog No. G2001601-1MG
n/a
Recombinant Human Basic Fibroblast Growth FactorRecombinant Human Basic Fibroblast Growth Factor
Recombinant Human Basic Fibroblast Growth Factor
$995.00 
Catalog No. G2001602-1MG
n/a
Recombinant Human Epidermal Growth FactorRecombinant Human Epidermal Growth Factor
Recombinant Human Epidermal Growth Factor
$140.00 
Catalog No. G2001603-1MG
n/a
Recombinant Human Insulin-like Growth Factor-1Recombinant Human Insulin-like Growth Factor-1
Recombinant Human Insulin-like Growth Factor-1
$235.00 
Catalog No. G2001604-1MG
n/a
Recombinant Human Plaet-Derived Growth Factor-BBRecombinant Human Plaet-Derived Growth Factor-BB
Recombinant Human Plaet-Derived Growth Factor-BB
$3200.00 
Catalog No. G2001605-1MG
n/a
Recombinant Human| Transforming Growth Factor,Beta 1Recombinant Human| Transforming Growth Factor,Beta 1
Recombinant Human| Transforming Growth Factor,Beta 1
$5050.00 
Catalog No. G2001606-1MG
n/a
Recombinant Mouse Basic Fibroblast Growth FactorRecombinant Mouse Basic Fibroblast Growth Factor
Recombinant Mouse Basic Fibroblast Growth Factor
$880.00 
Catalog No. G2001652-1MG
n/a
Recombinant Mouse Epidermal Growth FactorRecombinant Mouse Epidermal Growth Factor
Recombinant Mouse Epidermal Growth Factor
$220.00 
Catalog No. G2001653-1MG
n/a
Recombinant Mouse Leukemia Inhibitory FactorRecombinant Mouse Leukemia Inhibitory Factor
Recombinant Mouse Leukemia Inhibitory Factor
$2640.00 
Catalog No. G2001651-1MG
n/a
Remodelin, Acetyl-transferase NAT10 InhibitorRemodelin, Acetyl-transferase NAT10 Inhibitor
Remodelin, Acetyl-transferase NAT10 Inhibitor
$139.00 
Catalog No. M60187
Remodelin is a novel potent and selective inhibitor of the acetyl-transferase protein NAT10.
RepSox---TGF-β Type I Receptor ALK5 Inhibitor RepSox---TGF-β Type I Receptor ALK5 Inhibitor 
RepSox---TGF-β Type I Receptor ALK5 Inhibitor
$79.00 
Catalog No. M60151
RepSox (E-616452 or SJN 2511) is a highly potent, selective inhibitor of the TGF-β type I receptor ALK5.
RG108---DNA Methyltransferase InhibitorRG108---DNA Methyltransferase Inhibitor
RG108---DNA Methyltransferase Inhibitor
$65.00 
Catalog No. M60176
RG108 is a potent, selective and cell permeable inhibitor of DNA methyltransferase.
RG2833 (RGFP109), Brain-penetrant HDAC InhibitorRG2833 (RGFP109), Brain-penetrant HDAC Inhibitor
RG2833 (RGFP109), Brain-penetrant HDAC Inhibitor
$69.00 
Catalog No. M60225
A potent and selective brain-penetrant HDAC inhibitor HDAC1 and HDAC3.
RGFP966, HDAC3 Inhibitor RGFP966, HDAC3 Inhibitor 
RGFP966, HDAC3 Inhibitor
$89.00 
Catalog No. M60156
RGFP966 is a potent and selective HDAC3 inhibitor.
RN-1, LSD1 Inhibitor RN-1, LSD1 Inhibitor 
RN-1, LSD1 Inhibitor
$109.00 
Catalog No. M60169
RN-1 is a potent, specific and brain-penetrant Lysine Specific Demethylase-1 (LSD1) inhibitor.
RO4929097, γ-Secretase InhibitorRO4929097, γ-Secretase Inhibitor
RO4929097, γ-Secretase Inhibitor
$109.00 
Catalog No. M60007
A potent and selective γ-secretase inhibitor; inhibits Notch signaling in stem cells and tumor cells.
RS-1, CRISPR Editing Enhancer RS-1, CRISPR Editing Enhancer 
RS-1, CRISPR Editing Enhancer
$89.00 
Catalog No. M60300
Previously characterized as a RAD51-Stimulatory compound and now found to be an HDR enhancer to enhance CRISPR/Cas9- and TALEN-mediated knock-in efficiency
RU-SKI 43, Hhat InhibitorRU-SKI 43, Hhat Inhibitor
RU-SKI 43, Hhat Inhibitor
$139.00 
Catalog No. M60100
The first potent and specific small molecule inhibitor of Hedgehog acyltransferase (Hhat).
RVX-208, BET Bromodomain InhibitorRVX-208, BET Bromodomain Inhibitor
RVX-208, BET Bromodomain Inhibitor
$59.00 
Catalog No. M60177
RVX-208 is a potent and selective BET bromodomain inhibitor for the second bromodomain (BD2), ~170-fold selectivity over BD1.
Ryuvidine, Lysine Methyltransferase SETD8 InhibitorRyuvidine, Lysine Methyltransferase SETD8 Inhibitor
Ryuvidine, Lysine Methyltransferase SETD8 Inhibitor
$129.00 
Catalog No. M60252
A potent, selective and cell permeable lysine methyltransferase SETD8 inhibitor.
SAG, Hedgehog AgonistSAG, Hedgehog Agonist
SAG, Hedgehog Agonist
$129.00 
Catalog No. M60081
A potent, selective, and cell-permeable small-molecule agonist of the Hedgehog pathway.
SB431542, TGF-beta InhibitorSB431542, TGF-beta Inhibitor
SB431542, TGF-beta Inhibitor
$300.00 
Catalog No. M60015
A potent and selective TGF-β pathway inhibitor (selective for ALK4, ALK5 and ALK7).
SBI-0206965, Autophagy Kinase ULK1 InhibitorSBI-0206965, Autophagy Kinase ULK1 Inhibitor
SBI-0206965, Autophagy Kinase ULK1 Inhibitor
$129.00 
Catalog No. M60268
A potent, selective and cell permeable autophagy kinase ULK1 inhibitor.
SCH51344, MTH1 Inhibitor SCH51344, MTH1 Inhibitor 
SCH51344, MTH1 Inhibitor
$139.00 
Catalog No. M60212
A novel potent, selective and cell permeable MTH1 inhibitor.
SCR7, NHEJ inhibitorSCR7, NHEJ inhibitor
SCR7, NHEJ inhibitor
$129.00 
Catalog No. M60082
A potent and selective inhibitor of non-homologous end joining (NHEJ).
SD70, Histone Demethylase JMJD2  Inhibitor SD70, Histone Demethylase JMJD2  Inhibitor 
SD70, Histone Demethylase JMJD2 Inhibitor
$139.00 
Catalog No. M60194
A potent, selective and cell-permeable inhibitor of histone demethylase JMJD2 (KDM4C).
Sephin1, PPP1R1 Protein Phosphatase InhibitorSephin1, PPP1R1 Protein Phosphatase Inhibitor
Sephin1, PPP1R1 Protein Phosphatase Inhibitor
$129.00 
Catalog No. M60280
A potent, selective and bioavailable inhibitor of the regulatory subunit PPP1R1 of protein phosphatase 1.
SGC-CBP30, p300/CBP Bromodomain Inhibitor SGC-CBP30, p300/CBP Bromodomain Inhibitor 
SGC-CBP30, p300/CBP Bromodomain Inhibitor
$139.00 
Catalog No. M60138
SGC-CBP30 is a highly potent and selective p300/CBP bromodomain inhibitor
SGC0946, DOT1L inhibitor SGC0946, DOT1L inhibitor 
SGC0946, DOT1L inhibitor
$139.00 
Catalog No. M60101
A highly potent and selective inhibitor of DOT1L methyltransferase.
SGC707, Allosteric PRMT3 InhibitorSGC707, Allosteric PRMT3 Inhibitor
SGC707, Allosteric PRMT3 Inhibitor
$129.00 
Catalog No. M60243
A potent, selective and cell permeable allosteric protein arginine methyltransferase 3 (PRMT3) inhibitor.
SGI-1027, DNMT InhibitorSGI-1027, DNMT Inhibitor
SGI-1027, DNMT Inhibitor
$89.00 
Catalog No. M60155
A potent and selective inhibitor of DNA methyltransferase (DNMT).
SHP099, SHP2 Phosphatase InhibitorSHP099, SHP2 Phosphatase Inhibitor
SHP099, SHP2 Phosphatase Inhibitor
$139.00 
Catalog No. M60319
A highly potent, selective and orally bioavailable small-molecule SHP2 inhibitor.
SirReal2, Sirt2 InhibitorSirReal2, Sirt2 Inhibitor
SirReal2, Sirt2 Inhibitor
$119.00 
Catalog No. M60289
A potent and selective Sirt2 inhibitor.
SIRT1 Polyclonal AntibodySIRT1 Polyclonal Antibody
SIRT1 Polyclonal Antibody
$0.00 
Catalog No. A90007
SIRT1 Polyclonal Antibody: SIRT1 is a nuclear protein that regulates epigenetic gene silencing and suppresses recombination of rDNA
SKP2-C25, Skp2 InhibitorSKP2-C25, Skp2 Inhibitor
SKP2-C25, Skp2 Inhibitor
$139.00 
Catalog No. M60136
A potent, selective and cell permeable Skp2 inhibitor, selectively inhibits Skp2 E3 ligase activity, but not activity of other SCF complexes.
SKPin C1, Skp2 Inhibitor SKPin C1, Skp2 Inhibitor 
SKPin C1, Skp2 Inhibitor
$109.00 
Catalog No. M60137
A potent and selective inhibitor of Skp2-mediated p27 degradation.
SMER3, SCF family E3 Ubiquitin Ligase Inhibitor SMER3, SCF family E3 Ubiquitin Ligase Inhibitor 
SMER3, SCF family E3 Ubiquitin Ligase Inhibitor
$129.00 
Catalog No. M60250
A potent and selective a yeast SCF family E3 ubiquitin ligase inhibitor, also a small-molecule enhancers of rapamycin.
Spautin-1, Autophagy InhibitorSpautin-1, Autophagy Inhibitor
Spautin-1, Autophagy Inhibitor
$69.00 
Catalog No. M60003
A potent autophagy inhibitor, selectively promotes the degradation of Vps34 complexes.
SR10067, REV-ERB AgonistSR10067, REV-ERB Agonist
SR10067, REV-ERB Agonist
$129.00 
Catalog No. M60240
A potent and specific synthetic REV-ERB agonist.
SR1664,PPAR-γ ModulatorSR1664,PPAR-γ Modulator
SR1664,PPAR-γ Modulator
$109.00 
Catalog No. M66048
An unique PPARγ modulator that has potent anti-diabetic activity through blocking the Cdk5-mediated phosphorylation of PPARγ, but compley lacks classical transcriptional agonism that accounts for other PPARγ agonists’ side effects.
SR9009, REV-ERB AgonistSR9009, REV-ERB Agonist
SR9009, REV-ERB Agonist
$109.00 
Catalog No. M60236
A potent and specific synthetic REV-ERB agonist.
SR9011SR9011
SR9011
$1250.00 
Catalog No. M66049-b
SR9011, REV-ERB AgonistSR9011, REV-ERB Agonist
SR9011, REV-ERB Agonist
$109.00 
Catalog No. M66049
A potent synthetic REV-ERB agonist with in vivo activity; can regulate circadian behavior and metabolism.
SR9011-cSR9011-c
SR9011-c
$1250.00 
Catalog No. SR9011-c
SR9243, LXR Inverse AgonistSR9243, LXR Inverse Agonist
SR9243, LXR Inverse Agonist
$129.00 
Catalog No. M60270
A highly potent and selective small molecule LXR inverse agonist that induces LXR-corepressor interaction.
StemRegenin1 (SR1)---HSC Expansion MoleculeStemRegenin1 (SR1)---HSC Expansion Molecule
StemRegenin1 (SR1)---HSC Expansion Molecule
$99.00 
Catalog No. M60001
A potent and selective aryl hydrocarbon receptor antagonist; can promote robust expansion of human CD34+ hematopoietic stem and progenitor cells.
SU5402---FGFR inhibitor SU5402---FGFR inhibitor 
SU5402---FGFR inhibitor
$89.00 
Catalog No. M60025
A potent and selective inhibitor of FGFR, VEGFR, and PDGFR.
SW033291, 15-PGDH InhibitorSW033291, 15-PGDH Inhibitor
SW033291, 15-PGDH Inhibitor
$99.00 
Catalog No. M60298
A highly potent and selective inhibitor of 15-PGDH to increase prostaglandin PGE2 levels in bone marrow and other tissues.
TAK-875 (Fasiglifam), GPR40 AgonistTAK-875 (Fasiglifam), GPR40 Agonist
TAK-875 (Fasiglifam), GPR40 Agonist
$139.00 
Catalog No. M60220
A potent, selective and orally bioavailable partial GPR40 agonist.
TAME, Ubiquitin Ligase APC/C InhibitorTAME, Ubiquitin Ligase APC/C Inhibitor
TAME, Ubiquitin Ligase APC/C Inhibitor
$29.00 
Catalog No. M60246
A competitive inhibitor of the ubiquitin ligase anaphase-promoting complex/cyclosome (APC/C).
Tasquinimod, Allosteric HDAC4 InhibitorTasquinimod, Allosteric HDAC4 Inhibitor
Tasquinimod, Allosteric HDAC4 Inhibitor
$129.00 
Catalog No. M60235
A potent and selective allosteric HDAC4 inhibitor.
TCID, Ubiquitin C-terminal Hydrolase-L3 (UCH-L3) Inhibitor TCID, Ubiquitin C-terminal Hydrolase-L3 (UCH-L3) Inhibitor 
TCID, Ubiquitin C-terminal Hydrolase-L3 (UCH-L3) Inhibitor
$99.00 
Catalog No. M60197
A novel potent and selective inhibitor of ubiquitin C-terminal hydrolase-L3 (UCH-L3)
TEPP-46 (ML265), Pyruvate Kinase M2 (PKM2) ActivatorTEPP-46 (ML265), Pyruvate Kinase M2 (PKM2) Activator
TEPP-46 (ML265), Pyruvate Kinase M2 (PKM2) Activator
$129.00 
Catalog No. M60304
A potent and selective Pyruvate kinase M2 (PKM2) activator.
TG101348 (SAR302503), JAK2 and BRD4 Dual Inhibitor TG101348 (SAR302503), JAK2 and BRD4 Dual Inhibitor 
TG101348 (SAR302503), JAK2 and BRD4 Dual Inhibitor
$109.00 
Catalog No. M60172
TG101348 is a potent, specific and orally bioavailable inhibitor of JAK2 and BRD4 in clinical trials.
TH-302, Hypoxia-activated Pro-drugTH-302, Hypoxia-activated Pro-drug
TH-302, Hypoxia-activated Pro-drug
$179.00 
Catalog No. M60089
A highly potent and selective hypoxia-activated pro-drug targeting hypoxic regions of solid tumors.
TH588, MTH1 InhibitorTH588, MTH1 Inhibitor
TH588, MTH1 Inhibitor
$139.00 
Catalog No. M60211
A novel potent, selective and cell permeable MTH1 inhibitor.
Thiazovivin, Rock Inhibitor Thiazovivin, Rock Inhibitor 
Thiazovivin, Rock Inhibitor
$79.00 
Catalog No. M60009
A more potent and selective Rock inhibitor; can enhance hESC and hiPSC survival from single cell dissociation.
THZ1, Covalent CDK7 InhibitorTHZ1, Covalent CDK7 Inhibitor
THZ1, Covalent CDK7 Inhibitor
$159.00 
Catalog No. M60214
A novel potent, selective and cell permeable irreversible CDK7 inhibitor.
TMP269, Class IIa HDAC InhibitorTMP269, Class IIa HDAC Inhibitor
TMP269, Class IIa HDAC Inhibitor
$129.00 
Catalog No. M60119
A highly potent, selective and cell-permeable class IIa HDAC inhibitor.
TMPA---AMPK ActivatorTMPA---AMPK Activator
TMPA---AMPK Activator
$119.00 
Catalog No. M60072
TMPA is a novel small molecule that binds to orphan Nuclear Receptor Nur77 and activates AMPK.
TRIM24-C34, BRPF1B/TRIM24 Dual InhibitorTRIM24-C34, BRPF1B/TRIM24 Dual Inhibitor
TRIM24-C34, BRPF1B/TRIM24 Dual Inhibitor
$99.00 
Catalog No. M60265
A potent, selective and cell permeable BRPF1B and TRIM24 dual inhibitor.
TRIM24-C34bulkTRIM24-C34bulk
TRIM24-C34bulk
$169.00   $199.00 
Catalog No. M60265-b
TRIM24-C34bulkTRIM24-C34bulk
TRIM24-C34bulk
$0.00 
Catalog No. M60265-b
TZ9, Rad6 Ubiquitin Inhibitor TZ9, Rad6 Ubiquitin Inhibitor 
TZ9, Rad6 Ubiquitin Inhibitor
$109.00 
Catalog No. M60286
A selective and cell permeable inhibitor of human E2 ubiquitin-conjugating enzyme Rad6B.
UF010, HDAC InhibitorUF010, HDAC Inhibitor
UF010, HDAC Inhibitor
$89.00 
Catalog No. M60278
UF010 is a potent and selective class I HADC inhibitor.
UM171, Human HSC Self-renewal AgonistUM171, Human HSC Self-renewal Agonist
UM171, Human HSC Self-renewal Agonist
$159.00 
Catalog No. M60223
A potent small molecules that stimulates the expansion ex vivo of human cord blood cells capable of reconstituting human hematopoiesis for at least 6 months in immunocompromised mice.
UNC0379, Lysine Methyltransferase SETD8 Inhibitor UNC0379, Lysine Methyltransferase SETD8 Inhibitor 
UNC0379, Lysine Methyltransferase SETD8 Inhibitor
$129.00 
Catalog No. M60207
A novel selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8
UNC0638, G9a HMTase Inhibitor UNC0638, G9a HMTase Inhibitor 
UNC0638, G9a HMTase Inhibitor
$89.00 
Catalog No. M66056
A potent, selective and cell permeable inhibitor of G9a (EHMT2) and GLP (EHMT1) histone methyltransferases.
UNC0642, G9a/GLP HMTase Inhibitor UNC0642, G9a/GLP HMTase Inhibitor 
UNC0642, G9a/GLP HMTase Inhibitor
$129.00 
Catalog No. M60185
A novel highly potent, selective and cell permeable inhibitor of the homologous protein lysine methyltransferases, G9a and GLP, with improved PK properties.
UNC0646, G9a/GLP HMTase Inhibitor UNC0646, G9a/GLP HMTase Inhibitor 
UNC0646, G9a/GLP HMTase Inhibitor
$89.00 
Catalog No. M60184
A novel potent, selective and cell permeable homologous protein lysine methyltransferases G9a and GLP inhibitor.
UNC1215, L3MBTL3 Domain InhibitorUNC1215, L3MBTL3 Domain Inhibitor
UNC1215, L3MBTL3 Domain Inhibitor
$119.00 
Catalog No. M60084
A highly potent and selective small molecule inhibitor for the methyl-lysine (Kme) reading function of L3MBTL3.
UNC2170, Methyl-lysine Binding Protein 53BP1 InhibitorUNC2170, Methyl-lysine Binding Protein 53BP1 Inhibitor
UNC2170, Methyl-lysine Binding Protein 53BP1 Inhibitor
$99.00 
Catalog No. M60260
A selective and cell permeable methyl-lysine binding protein 53BP1 antagonist.
UNC2327, Allosteric PRMT3 Inhibitor UNC2327, Allosteric PRMT3 Inhibitor 
UNC2327, Allosteric PRMT3 Inhibitor
$129.00 
Catalog No. M60253
A potent and selective allosteric protein arginine methyltransferase 3 (PRMT3) inhibitor.
UNC669, L3MBTL1 Domain Inhibitor UNC669, L3MBTL1 Domain Inhibitor 
UNC669, L3MBTL1 Domain Inhibitor
$89.00 
Catalog No. M60083
A potent and selective small molecule inhibitor for the methyl-lysine (Kme) reading function of L3MBTL1
Verteporfin (Visudyne), YAP InhibitorVerteporfin (Visudyne), YAP Inhibitor
Verteporfin (Visudyne), YAP Inhibitor
$59.00 
Catalog No. M60247
A potent and selective YAP inhibitor to disrupt YAP-TEAD interactions and enhance trypsin cleavage of YAP.
VLX600, Mitochondrial OXPHOS InhibitorVLX600, Mitochondrial OXPHOS Inhibitor
VLX600, Mitochondrial OXPHOS Inhibitor
$69.00 
Catalog No. M60261
A potent and selective mitochondrial OXPHOS inhibitor.
VR23, Proteasome InhibitorVR23, Proteasome Inhibitor
VR23, Proteasome Inhibitor
$99.00 
Catalog No. M60307
A potent and selective proteasome inhibitor with IC50 of 1 nM, 50-100 nM, and 3 μM for trypsin-like proteasomes, chymotrypsin-like proteasomes,
WAY-316606, Secreted Frizzled-related Protein-1 (sFRP-1) Inhibitor WAY-316606, Secreted Frizzled-related Protein-1 (sFRP-1) Inhibitor 
WAY-316606, Secreted Frizzled-related Protein-1 (sFRP-1) Inhibitor
$139.00 
Catalog No. M60215
A novel potent and selective inhibitor of secreted frizzled-related protein-1 (sFRP-1) to increase Wnt signaling.
WDR5-0103, WDR5 InhibitorWDR5-0103, WDR5 Inhibitor
WDR5-0103, WDR5 Inhibitor
$89.00 
Catalog No. M60233
A potent and selective WD repeat-containing protein 5 (WDR5) antagonist.
WDR5-C47, WDR5-MLL (SET1) Antagonist WDR5-C47, WDR5-MLL (SET1) Antagonist 
WDR5-C47, WDR5-MLL (SET1) Antagonist
$129.00 
Catalog No. M60118
A highly potent and selective antagonist of WDR5-MLL interaction.
Wnt-C59, Wnt Antagonist Wnt-C59, Wnt Antagonist 
Wnt-C59, Wnt Antagonist
$89.00 
Catalog No. M60005
A potent, selective and oral active Wnt  signaling pathway antagonist.
WP1130 (Degrasyn), Deubiquitinylating Enzyme (DUB) Inhibitor WP1130 (Degrasyn), Deubiquitinylating Enzyme (DUB) Inhibitor 
WP1130 (Degrasyn), Deubiquitinylating Enzyme (DUB) Inhibitor
$69.00 
Catalog No. M60206
A cell-permeable, potent and selective inhibitor of the deubiquitinylating enzymes (DUBs).
WS3, β Cell Proliferation Inducer WS3, β Cell Proliferation Inducer 
WS3, β Cell Proliferation Inducer
$139.00 
Catalog No. M60095
A highly potent and selective small molecule that promotes pancreatic β cell and RPE cells expansion.
WS6, β Cell Proliferation Inducer WS6, β Cell Proliferation Inducer 
WS6, β Cell Proliferation Inducer
$139.00 
Catalog No. M60097
A highly potent and selective small molecule that promotes pancreatic β cell proliferation in rodent and human primary islets and shows excellent in vivo efficacy.
WWL113, Ces3 and Ces1f Inhibitor WWL113, Ces3 and Ces1f Inhibitor 
WWL113, Ces3 and Ces1f Inhibitor
$139.00 
Catalog No. M60162
A novel potent and selective inhibitor of Ces3 and Ces1f
XAV939---Wnt Antagonist XAV939---Wnt Antagonist 
XAV939---Wnt Antagonist
$89.00 
Catalog No. M60010
A potent and selective Wnt pathway antagonist; functions to stabilize axin by inhibiting tankyrase 1 and tankyrase 2.
XL888---HSP90 InhibitorXL888---HSP90 Inhibitor
XL888---HSP90 Inhibitor
$149.00 
Catalog No. M60164
A highly potent, ATP-competitive and orally bioavailable Hsp90 inhibitor.
Y-27632---Rock Inhibitor Y-27632---Rock Inhibitor 
Y-27632---Rock Inhibitor
$69.00 
Catalog No. M60011
The most widely used Rock kinase inhibitor.
Y-320---IL-17 ImmunomodulatorY-320---IL-17 Immunomodulator
Y-320---IL-17 Immunomodulator
$89.00 
Catalog No. M60200
An orally active potent immunomodulator, inhibits IL-15-induced IL-17 production by CD4 T cells.
ZCL278---Cdc42 GTPase InhibitorZCL278---Cdc42 GTPase Inhibitor
ZCL278---Cdc42 GTPase Inhibitor
$119.00 
Catalog No. M60133
A potent and selective inhibitor of Cdc42 GTPase.
ZLN005---PGC-1α Transcriptional ActivatorZLN005---PGC-1α Transcriptional Activator
ZLN005---PGC-1α Transcriptional Activator
$69.00 
Catalog No. M60142  
A potent and selective small molecule PGC-1α transcriptional activator.